MLN-8054 KINOMEscan - Dataset (ID:20157)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200167 VGFR1 200167 P17948
Vascular endothelial growth factor receptor 1; fms-related tyrosine kinase 1; vascular permeability factor receptor; FLT; FLT1; VEGFR1
KINOMEscan Wild Type; Partial length
200168 FLT3 200168 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan Wild Type; Partial length
200175 FLT4 200175 P35916
Fms-related tyrosine kinase 4; FLT4; FLT41; LMPH1A; PCL; VEGFR3
KINOMEscan Wild Type; Partial length
200176 FRK 200176 P42685
Tyrosine-protein kinase FRK; Fyn-related kinase; FRK; GTK; PTK5; RAK
KINOMEscan Wild Type; Partial length
200177 FYN 200177 P06241
FYN oncogene related to SRC, FGR, YES; FYN; MGC45350; SLK; SYN
KINOMEscan Wild Type; Partial length
200178 GAK 200178 O14976
Cyclin G associated kinase; FLJ16629; FLJ40395; GAK; MGC99654
KINOMEscan Wild Type; Partial length
200179 GCN2(Kin.Dom.2,S808G) 200179 Q9P2K8
Eukaryotic translation initiation factor 2 alpha kinase 4; EIF2AK4; GCN2; KIAA1338
KINOMEscan S808G Kin.Dom.2 Wild Type; Partial length
200186 HIPK1 200186 Q86Z02
Homeodomain interacting protein kinase 1; HIPK1; KIAA0630; MGC26642; MGC33446; MGC33548; Myak; Nbak2
KINOMEscan Wild Type; Partial length
200187 HIPK2 200187 Q9H2X6
Homeodomain interacting protein kinase 2; DKFZp686K02111; FLJ23711; HIPK2; PRO0593
KINOMEscan Wild Type; Partial length
200188 HIPK3 200188 Q9H422
Homeodomain interacting protein kinase 3; DYRK6; FIST3; HIPK3; PKY; YAK1
KINOMEscan Wild Type; Partial length
200189 HIPK4 200189 Q8NE63
Homeodomain interacting protein kinase 4; FLJ32818; HIPK4
KINOMEscan Wild Type; Partial length
200191 HUNK 200191 P57058
Hormonally up-regulated Neu-associated kinase; HUNK
KINOMEscan Wild Type; Partial length
200192 ICK 200192 Q9UPZ9
Intestinal cell (MAK-like) kinase; ECO; ICK; KIAA0936; LCK2; MGC46090; MRK
KINOMEscan Wild Type; Partial length
200193 IGF1R 200193 P08069
Insulin-like growth factor 1 receptor; CD221; IGF1R; IGFIR; IGFR; JTK13; MGC142170; MGC142172; MGC18216
KINOMEscan Wild Type; Partial length
200197 INSR 200197 P06213
Insulin receptor; CD220; HHF5; INSR; IR
KINOMEscan Wild Type; Partial length
200198 INSRR 200198 P14616
Insulin receptor-related receptor; INSRR; IRR
KINOMEscan Wild Type; Partial length
200199 IRAK1 200199 P51617
Interleukin-1 receptor-associated kinase 1
KINOMEscan Wild Type; Partial length
200200 IRAK3 200200 Q9Y616
Interleukin-1 receptor-associated kinase 3; ASRT5; FLJ13601; IRAK3; IRAKM
KINOMEscan Wild Type; Partial length
200201 IRAK4 200201 Q9NWZ3
Interleukin-1 receptor-associated kinase 4; IPD1; NY-REN-64; REN64
KINOMEscan Wild Type; Partial length
200202 ITK 200202 Q08881
IL2-inducible T-cell kinase; EMT; ITK; LYK; MGC126257; MGC126258; PSCTK2
KINOMEscan Wild Type; Partial length
200203 JAK1(JH1domain-catalytic) 200203 P23458
Janus kinase 1; JAK1; JAK1A; JAK1B; JAK1-catalytic; JTK3
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200204 JAK1(JH2domain-pseudokinase) 200204 P23458
Janus kinase 1; JAK1; JAK1~b; JAK1A; JAK1B; JAK1-pseudokinase; JTK3
KINOMEscan JH2domain-pseudokinase Wild Type; Partial length
200207 JAK2(JH1domain-catalytic) 200207 O60674
Janus kinase 2; JAK2; JAK2-catalytic; JTK10
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200209 JAK3(JH1domain-catalytic) 200209 P52333
Tyrosine-protein kinase JAK3; Janus kinase 3; JAK-3; L-JAK
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200213 JNK3 200213 P53779
Mitogen-activated protein kinase 10; FLJ12099; FLJ33785; JNK3; JNK3A; MAPK10; MGC50974; p493F12; p54bSAPK; PRKM10
KINOMEscan Wild Type; Partial length