AZD-6244 KINOMEscan - Dataset (ID:20156)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Selumetinib | FES | nM | |
Selumetinib | FGFR1 | nM | |
Selumetinib | FGFR2 | nM | |
Selumetinib | FGFR3 | nM | |
Selumetinib | FGFR3(G697C) | nM | |
Selumetinib | FGFR4 | nM | |
Selumetinib | FGR | nM | |
Selumetinib | VGFR1 | nM | |
Selumetinib | FLT3 | nM | |
Selumetinib | FLT3(D835H) | nM | |
Selumetinib | FLT3(D835Y) | nM | |
Selumetinib | FLT3(ITD) | nM | |
Selumetinib | FLT3(K663Q) | nM | |
Selumetinib | FLT3(N841I) | nM | |
Selumetinib | FLT3(R834Q) | nM | |
Selumetinib | FLT4 | nM | |
Selumetinib | FRK | nM | |
Selumetinib | FYN | nM | |
Selumetinib | GAK | nM | |
Selumetinib | GCN2(Kin.Dom.2,S808G) | nM | |
Selumetinib | GRK1 | nM | |
Selumetinib | GRK4 | nM | |
Selumetinib | GRK7 | nM | |
Selumetinib | GSK3A | nM | |
Selumetinib | GSK3B | nM |