PLX-4720 KINOMEscan-2 - Dataset (ID:20154)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PLX-4720 | FES | 3600.0 | nM |
PLX-4720 | FGFR1 | 5300.0 | nM |
PLX-4720 | FGFR2 | 3100.0 | nM |
PLX-4720 | FGFR3 | nM | |
PLX-4720 | FGFR3(G697C) | nM | |
PLX-4720 | FGFR4 | nM | |
PLX-4720 | FGR | 62.0 | nM |
PLX-4720 | VGFR1 | 1900.0 | nM |
PLX-4720 | FLT3 | 1300.0 | nM |
PLX-4720 | FLT3(D835H) | 6100.0 | nM |
PLX-4720 | FLT3(D835Y) | 6500.0 | nM |
PLX-4720 | FLT3(ITD) | 6100.0 | nM |
PLX-4720 | FLT3(K663Q) | 2300.0 | nM |
PLX-4720 | FLT3(N841I) | 3900.0 | nM |
PLX-4720 | FLT3(R834Q) | 3000.0 | nM |
PLX-4720 | FLT4 | nM | |
PLX-4720 | FRK | 1900.0 | nM |
PLX-4720 | FYN | 2300.0 | nM |
PLX-4720 | GAK | nM | |
PLX-4720 | GCN2(Kin.Dom.2,S808G) | 1300.0 | nM |
PLX-4720 | GRK1 | nM | |
PLX-4720 | GRK4 | nM | |
PLX-4720 | GRK7 | nM | |
PLX-4720 | GSK3A | nM | |
PLX-4720 | GSK3B | nM |