PLX-4720 KINOMEscan-2 - Dataset (ID:20154)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PLX-4720 | EPHB6 | 860.0 | nM |
PLX-4720 | TGFBR2 | 890.0 | nM |
PLX-4720 | ABL1(F317L)-nonphosphorylated | 940.0 | nM |
PLX-4720 | MP2K2 | 1100.0 | nM |
PLX-4720 | LYN | 1100.0 | nM |
PLX-4720 | BLK | 1100.0 | nM |
PLX-4720 | TNK2 | 1100.0 | nM |
PLX-4720 | PIK4CB | 1200.0 | nM |
PLX-4720 | FLT3 | 1300.0 | nM |
PLX-4720 | ABL1(F317I)-nonphosphorylated | 1300.0 | nM |
PLX-4720 | GCN2(Kin.Dom.2,S808G) | 1300.0 | nM |
PLX-4720 | PAK1 | 1400.0 | nM |
PLX-4720 | TESK1 | 1500.0 | nM |
PLX-4720 | LCK | 1800.0 | nM |
PLX-4720 | YES | 1800.0 | nM |
PLX-4720 | ABL1(Y253F)-phosphorylated | 1900.0 | nM |
PLX-4720 | SIK2 | 1900.0 | nM |
PLX-4720 | VGFR1 | 1900.0 | nM |
PLX-4720 | FRK | 1900.0 | nM |
PLX-4720 | CDK8 | 1900.0 | nM |
PLX-4720 | CAMK1 | 1900.0 | nM |
PLX-4720 | STK16 | 1900.0 | nM |
PLX-4720 | VGFR2 | 2100.0 | nM |
PLX-4720 | CSK | 2200.0 | nM |
PLX-4720 | FLT3(K663Q) | 2300.0 | nM |