PLX-4720 KINOMEscan-2 - Dataset (ID:20154)

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Small Molecule Protein Kd Conc unit
PLX-4720 EPHB6 860.0
nM
PLX-4720 TGFBR2 890.0
nM
PLX-4720 ABL1(F317L)-nonphosphorylated 940.0
nM
PLX-4720 MP2K2 1100.0
nM
PLX-4720 LYN 1100.0
nM
PLX-4720 BLK 1100.0
nM
PLX-4720 TNK2 1100.0
nM
PLX-4720 PIK4CB 1200.0
nM
PLX-4720 FLT3 1300.0
nM
PLX-4720 ABL1(F317I)-nonphosphorylated 1300.0
nM
PLX-4720 GCN2(Kin.Dom.2,S808G) 1300.0
nM
PLX-4720 PAK1 1400.0
nM
PLX-4720 TESK1 1500.0
nM
PLX-4720 LCK 1800.0
nM
PLX-4720 YES 1800.0
nM
PLX-4720 ABL1(Y253F)-phosphorylated 1900.0
nM
PLX-4720 SIK2 1900.0
nM
PLX-4720 VGFR1 1900.0
nM
PLX-4720 FRK 1900.0
nM
PLX-4720 CDK8 1900.0
nM
PLX-4720 CAMK1 1900.0
nM
PLX-4720 STK16 1900.0
nM
PLX-4720 VGFR2 2100.0
nM
PLX-4720 CSK 2200.0
nM
PLX-4720 FLT3(K663Q) 2300.0
nM