GDC-0941 KINOMEscan-2 - Dataset (ID:20152)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pictilisib | FES | nM | |
Pictilisib | FGFR1 | nM | |
Pictilisib | FGFR2 | nM | |
Pictilisib | FGFR3 | nM | |
Pictilisib | FGFR3(G697C) | nM | |
Pictilisib | FGFR4 | nM | |
Pictilisib | FGR | nM | |
Pictilisib | VGFR1 | nM | |
Pictilisib | FLT3 | 2600.0 | nM |
Pictilisib | FLT3(D835H) | 1700.0 | nM |
Pictilisib | FLT3(D835Y) | 710.0 | nM |
Pictilisib | FLT3(ITD) | 2200.0 | nM |
Pictilisib | FLT3(K663Q) | 2600.0 | nM |
Pictilisib | FLT3(N841I) | 3900.0 | nM |
Pictilisib | FLT3(R834Q) | nM | |
Pictilisib | FLT4 | nM | |
Pictilisib | FRK | nM | |
Pictilisib | FYN | nM | |
Pictilisib | GAK | 2700.0 | nM |
Pictilisib | GCN2(Kin.Dom.2,S808G) | nM | |
Pictilisib | GRK1 | nM | |
Pictilisib | GRK4 | nM | |
Pictilisib | GRK7 | nM | |
Pictilisib | GSK3A | nM | |
Pictilisib | GSK3B | nM |