GDC-0941 KINOMEscan-2 - Dataset (ID:20152)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pictilisib | DCAMKL2 | nM | |
Pictilisib | DCAMKL3 | nM | |
Pictilisib | DDR1 | nM | |
Pictilisib | DDR2 | nM | |
Pictilisib | M3K12 | nM | |
Pictilisib | DMPK | nM | |
Pictilisib | DMPK2 | nM | |
Pictilisib | DRAK1 | nM | |
Pictilisib | DRAK2 | nM | |
Pictilisib | DYRK1A | nM | |
Pictilisib | DYRK1B | 3800.0 | nM |
Pictilisib | DYRK2 | 7600.0 | nM |
Pictilisib | EGFR | nM | |
Pictilisib | EGFR(E746-A750del) | nM | |
Pictilisib | EGFR(G719C) | nM | |
Pictilisib | EGFR(G719S) | nM | |
Pictilisib | EGFR(L747-E749del, A750P) | nM | |
Pictilisib | EGFR(L747-S752del, P753S) | nM | |
Pictilisib | EGFR(L747-T751del,Sins) | nM | |
Pictilisib | EGFR(L858R) | nM | |
Pictilisib | EGFR(L858R,T790M) | nM | |
Pictilisib | EGFR(L861Q) | nM | |
Pictilisib | EGFR(S752-I759del) | nM | |
Pictilisib | EGFR(T790M) | nM | |
Pictilisib | EIF2AK1 | nM |