BIRB-796 KINOMEscan - Dataset (ID:20151)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Doramapimod | CDK7 | 3100.0 | nM |
Doramapimod | FLT3(ITD) | 3000.0 | nM |
Doramapimod | ERK8 | 3000.0 | nM |
Doramapimod | EPHA4 | 2900.0 | nM |
Doramapimod | LYN | 2700.0 | nM |
Doramapimod | BRAF | 2700.0 | nM |
Doramapimod | KIT(V559D,V654A) | 2400.0 | nM |
Doramapimod | EGFR(T790M) | 2400.0 | nM |
Doramapimod | FLT3 | 2300.0 | nM |
Doramapimod | CIT | 2100.0 | nM |
Doramapimod | EPHA6 | 2000.0 | nM |
Doramapimod | CDK5 | 2000.0 | nM |
Doramapimod | MUSK | 1900.0 | nM |
Doramapimod | MKNK2 | 1600.0 | nM |
Doramapimod | EPHA5 | 1400.0 | nM |
Doramapimod | KIT(A829P) | 1400.0 | nM |
Doramapimod | LTK | 1400.0 | nM |
Doramapimod | ABL1(F317L)-nonphosphorylated | 1300.0 | nM |
Doramapimod | ABL2 | 1300.0 | nM |
Doramapimod | LCK | 1200.0 | nM |
Doramapimod | DMPK2 | 1200.0 | nM |
Doramapimod | FRK | 1200.0 | nM |
Doramapimod | PGFRA | 1200.0 | nM |
Doramapimod | PGFRB | 1100.0 | nM |
Doramapimod | CDC2L5 | 1100.0 | nM |