BIRB-796 KINOMEscan - Dataset (ID:20151)

The small molecule associated with this KINOMEscan dataset was erroneously assigned as HMS LINCS ID 10044-101 at the time of data release. The assignment was corrected to HMS LINCS 10169-999 on 2016-06-03.

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Small Molecule Protein Kd Conc unit
Doramapimod CDK7 3100.0
nM
Doramapimod FLT3(ITD) 3000.0
nM
Doramapimod ERK8 3000.0
nM
Doramapimod EPHA4 2900.0
nM
Doramapimod LYN 2700.0
nM
Doramapimod BRAF 2700.0
nM
Doramapimod KIT(V559D,V654A) 2400.0
nM
Doramapimod EGFR(T790M) 2400.0
nM
Doramapimod FLT3 2300.0
nM
Doramapimod CIT 2100.0
nM
Doramapimod EPHA6 2000.0
nM
Doramapimod CDK5 2000.0
nM
Doramapimod MUSK 1900.0
nM
Doramapimod MKNK2 1600.0
nM
Doramapimod EPHA5 1400.0
nM
Doramapimod KIT(A829P) 1400.0
nM
Doramapimod LTK 1400.0
nM
Doramapimod ABL1(F317L)-nonphosphorylated 1300.0
nM
Doramapimod ABL2 1300.0
nM
Doramapimod LCK 1200.0
nM
Doramapimod DMPK2 1200.0
nM
Doramapimod FRK 1200.0
nM
Doramapimod PGFRA 1200.0
nM
Doramapimod PGFRB 1100.0
nM
Doramapimod CDC2L5 1100.0
nM