AMG-706 KINOMEscan - Dataset (ID:20150)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Motesanib | FES | nM | |
| Motesanib | FGFR1 | 6200.0 | nM |
| Motesanib | FGFR2 | nM | |
| Motesanib | FGFR3 | nM | |
| Motesanib | FGFR3(G697C) | nM | |
| Motesanib | FGFR4 | 6800.0 | nM |
| Motesanib | FGR | 6900.0 | nM |
| Motesanib | VGFR1 | 12.0 | nM |
| Motesanib | FLT3 | 71.0 | nM |
| Motesanib | FLT3(D835H) | 4500.0 | nM |
| Motesanib | FLT3(D835Y) | 9500.0 | nM |
| Motesanib | FLT3(ITD) | 1000.0 | nM |
| Motesanib | FLT3(K663Q) | 54.0 | nM |
| Motesanib | FLT3(N841I) | 1100.0 | nM |
| Motesanib | FLT3(R834Q) | 3800.0 | nM |
| Motesanib | FLT4 | 9.7 | nM |
| Motesanib | FRK | 99.0 | nM |
| Motesanib | FYN | 2800.0 | nM |
| Motesanib | GAK | nM | |
| Motesanib | GCN2(Kin.Dom.2,S808G) | 4400.0 | nM |
| Motesanib | GRK1 | nM | |
| Motesanib | GRK4 | nM | |
| Motesanib | GRK7 | nM | |
| Motesanib | GSK3A | nM | |
| Motesanib | GSK3B | nM |