AMG-706 KINOMEscan - Dataset (ID:20150)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Motesanib | PRKX | nM | |
Motesanib | PRP4 | nM | |
Motesanib | FAK2 | nM | |
Motesanib | SIK3 | nM | |
Motesanib | RAF1 | 880.0 | nM |
Motesanib | RET | 14.0 | nM |
Motesanib | RET(M918T) | 20.0 | nM |
Motesanib | RET(V804L) | nM | |
Motesanib | RET(V804M) | nM | |
Motesanib | RIOK1 | nM | |
Motesanib | RIOK2 | nM | |
Motesanib | RIOK3 | nM | |
Motesanib | RIPK1 | nM | |
Motesanib | RIPK2 | 9300.0 | nM |
Motesanib | RIPK4 | nM | |
Motesanib | RIPK5 | nM | |
Motesanib | ROCK1 | nM | |
Motesanib | ROCK2 | nM | |
Motesanib | ROS1 | nM | |
Motesanib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
Motesanib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Motesanib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
Motesanib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Motesanib | RSK1(Kin.Dom.1-N-terminal) | nM | |
Motesanib | RSK1(Kin.Dom.2-C-terminal) | nM |