AMG-706 KINOMEscan - Dataset (ID:20150)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Motesanib | HIPK1 | nM | |
Motesanib | HIPK2 | nM | |
Motesanib | HIPK3 | nM | |
Motesanib | HIPK4 | nM | |
Motesanib | M4K1 | nM | |
Motesanib | HUNK | nM | |
Motesanib | ICK | nM | |
Motesanib | IGF1R | nM | |
Motesanib | IKKA | nM | |
Motesanib | IKKB | nM | |
Motesanib | IKKE | nM | |
Motesanib | INSR | nM | |
Motesanib | INSRR | nM | |
Motesanib | IRAK1 | nM | |
Motesanib | IRAK3 | nM | |
Motesanib | IRAK4 | nM | |
Motesanib | ITK | nM | |
Motesanib | JAK1(JH1domain-catalytic) | 5200.0 | nM |
Motesanib | JAK1(JH2domain-pseudokinase) | nM | |
Motesanib | JAK2(JH1domain-catalytic) | nM | |
Motesanib | JAK3(JH1domain-catalytic) | nM | |
Motesanib | JNK1 | nM | |
Motesanib | MK09 | nM | |
Motesanib | JNK3 | nM | |
Motesanib | AAK1 | nM |