BI-2536 KINOMEscan-2 - Dataset (ID:20149)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
BI-2536 | EGFR(G719C) | 630.0 | nM |
BI-2536 | RSK3(Kin.Dom.2-C-terminal) | 700.0 | nM |
BI-2536 | NEK3 | 720.0 | nM |
BI-2536 | NIM1 | 770.0 | nM |
BI-2536 | GRK7 | 850.0 | nM |
BI-2536 | DAPK2 | 930.0 | nM |
BI-2536 | CLK1 | 940.0 | nM |
BI-2536 | STK16 | 1100.0 | nM |
BI-2536 | STK33 | 1100.0 | nM |
BI-2536 | EGFR(L747-E749del, A750P) | 1100.0 | nM |
BI-2536 | JNK3 | 1100.0 | nM |
BI-2536 | LTK | 1200.0 | nM |
BI-2536 | CAMK2G | 1200.0 | nM |
BI-2536 | EGFR(L858R) | 1300.0 | nM |
BI-2536 | EGFR(G719S) | 1300.0 | nM |
BI-2536 | RSK4(Kin.Dom.2-C-terminal) | 1300.0 | nM |
BI-2536 | CAMK2A | 1300.0 | nM |
BI-2536 | CSNK1D | 1500.0 | nM |
BI-2536 | MINK | 1600.0 | nM |
BI-2536 | PHKG2 | 1600.0 | nM |
BI-2536 | TAOK3 | 1700.0 | nM |
BI-2536 | FES | 1900.0 | nM |
BI-2536 | EGFR(E746-A750del) | 1900.0 | nM |
BI-2536 | IRAK1 | 1900.0 | nM |
BI-2536 | CDK4-cyclinD3 | 1900.0 | nM |