BI-2536 KINOMEscan-2 - Dataset (ID:20149)

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Small Molecule Protein Kd Conc unit
BI-2536 EGFR(G719C) 630.0
nM
BI-2536 RSK3(Kin.Dom.2-C-terminal) 700.0
nM
BI-2536 NEK3 720.0
nM
BI-2536 NIM1 770.0
nM
BI-2536 GRK7 850.0
nM
BI-2536 DAPK2 930.0
nM
BI-2536 CLK1 940.0
nM
BI-2536 STK16 1100.0
nM
BI-2536 STK33 1100.0
nM
BI-2536 EGFR(L747-E749del, A750P) 1100.0
nM
BI-2536 JNK3 1100.0
nM
BI-2536 LTK 1200.0
nM
BI-2536 CAMK2G 1200.0
nM
BI-2536 EGFR(L858R) 1300.0
nM
BI-2536 EGFR(G719S) 1300.0
nM
BI-2536 RSK4(Kin.Dom.2-C-terminal) 1300.0
nM
BI-2536 CAMK2A 1300.0
nM
BI-2536 CSNK1D 1500.0
nM
BI-2536 MINK 1600.0
nM
BI-2536 PHKG2 1600.0
nM
BI-2536 TAOK3 1700.0
nM
BI-2536 FES 1900.0
nM
BI-2536 EGFR(E746-A750del) 1900.0
nM
BI-2536 IRAK1 1900.0
nM
BI-2536 CDK4-cyclinD3 1900.0
nM