R406 KINOMEscan-2 - Dataset (ID:20148)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
R406 | IKKB | 71.0 | nM |
R406 | IKKE | 13.0 | nM |
R406 | INSR | 1100.0 | nM |
R406 | INSRR | 4600.0 | nM |
R406 | IRAK1 | 9.7 | nM |
R406 | IRAK3 | 11.0 | nM |
R406 | IRAK4 | 140.0 | nM |
R406 | ITK | 400.0 | nM |
R406 | JAK1(JH1domain-catalytic) | 21.0 | nM |
R406 | JAK1(JH2domain-pseudokinase) | nM | |
R406 | JAK2(JH1domain-catalytic) | 3.5 | nM |
R406 | JAK3(JH1domain-catalytic) | 36.0 | nM |
R406 | JNK1 | 38.0 | nM |
R406 | JNK3 | 37.0 | nM |
R406 | KC1G1 | nM | |
R406 | KC1G2 | nM | |
R406 | KCC2D | 3000.0 | nM |
R406 | KCC4 | nM | |
R406 | KGP1 | nM | |
R406 | KGP2 | 3600.0 | nM |
R406 | KIT | 6.8 | nM |
R406 | KIT(A829P) | 3.5 | nM |
R406 | KIT(D816H) | 6.5 | nM |
R406 | KIT(D816V) | 2.5 | nM |
R406 | KIT(L576P) | 5.6 | nM |