R406 KINOMEscan-2 - Dataset (ID:20148)

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Small Molecule Protein Kd Conc unit
R406 TESK1 360.0
nM
R406 EPHA3 360.0
nM
R406 TLK2 380.0
nM
R406 BRAF(V600E) 380.0
nM
R406 MK12 390.0
nM
R406 ABL1(M351T)-phosphorylated 390.0
nM
R406 EPHB1 390.0
nM
R406 ABL1(H396P)-phosphorylated 390.0
nM
R406 ITK 400.0
nM
R406 SRPK3 400.0
nM
R406 AAK1 410.0
nM
R406 KIT(V559D,V654A) 410.0
nM
R406 ABL1(Q252H)-phosphorylated 430.0
nM
R406 CIT 440.0
nM
R406 EGFR(S752-I759del) 450.0
nM
R406 GRK4 450.0
nM
R406 CAMK1G 460.0
nM
R406 DYRK2 470.0
nM
R406 MST1R 470.0
nM
R406 MP2K6 480.0
nM
R406 TLK1 490.0
nM
R406 RSK1(Kin.Dom.1-N-terminal) 490.0
nM
R406 TAOK1 490.0
nM
R406 PKAC-beta 510.0
nM
R406 ABL1-nonphosphorylated 530.0
nM