AC220 KINOMEscan - Dataset (ID:20147)

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Small Molecule Protein Kd Conc unit
AC220 IKKB
nM
AC220 IKKE
nM
AC220 INSR
nM
AC220 INSRR
nM
AC220 IRAK1
nM
AC220 IRAK3
nM
AC220 IRAK4
nM
AC220 ITK
nM
AC220 JAK1(JH1domain-catalytic)
nM
AC220 JAK1(JH2domain-pseudokinase)
nM
AC220 JAK2(JH1domain-catalytic)
nM
AC220 JAK3(JH1domain-catalytic)
nM
AC220 JNK1
nM
AC220 JNK3
nM
AC220 KC1G1
nM
AC220 KC1G2
nM
AC220 KCC2D
nM
AC220 KCC4
nM
AC220 KGP1
nM
AC220 KGP2
nM
AC220 KIT 4.8
nM
AC220 KIT(A829P) 3.6
nM
AC220 KIT(D816H) 320.0
nM
AC220 KIT(D816V) 150.0
nM
AC220 KIT(L576P) 6.3
nM