AC220 KINOMEscan - Dataset (ID:20147)

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Small Molecule Protein Kd Conc unit
AC220 FLT3(D835H) 3.7
nM
AC220 FLT3(D835Y) 7.1
nM
AC220 FLT3(ITD) 8.8
nM
AC220 FLT3(K663Q) 2.2
nM
AC220 FLT3(N841I) 4.1
nM
AC220 FLT3(R834Q) 5.1
nM
AC220 FLT4 41.0
nM
AC220 FRK 1800.0
nM
AC220 FYN
nM
AC220 GAK
nM
AC220 GCN2(Kin.Dom.2,S808G)
nM
AC220 GRK1
nM
AC220 GRK4
nM
AC220 GRK7
nM
AC220 GSK3A
nM
AC220 GSK3B
nM
AC220 HCK
nM
AC220 HIPK1
nM
AC220 HIPK2
nM
AC220 HIPK3
nM
AC220 HIPK4 320.0
nM
AC220 HUNK
nM
AC220 ICK
nM
AC220 IGF1R
nM
AC220 IKKA
nM