AC220 KINOMEscan - Dataset (ID:20147)

Filter results: >>>>
Small Molecule Protein Kd Conc unit
AC220 HIPK4 320.0
nM
AC220 KIT(D816H) 320.0
nM
AC220 ERK8 270.0
nM
AC220 KIT(D816V) 150.0
nM
AC220 VGFR2 87.0
nM
AC220 DDR1 81.0
nM
AC220 FLT4 41.0
nM
AC220 VGFR1 41.0
nM
AC220 KIT(V559D,V654A) 36.0
nM
AC220 RET(V804L) 13.0
nM
AC220 PGFRA 11.0
nM
AC220 CSF1R 10.0
nM
AC220 RET(V804M) 9.1
nM
AC220 FLT3(ITD) 8.8
nM
AC220 RET 8.0
nM
AC220 PGFRB 7.7
nM
AC220 FLT3(D835Y) 7.1
nM
AC220 KIT(L576P) 6.3
nM
AC220 KIT(V559D,T670I) 6.0
nM
AC220 FLT3(R834Q) 5.1
nM
AC220 KIT(V559D) 5.0
nM
AC220 KIT 4.8
nM
AC220 FLT3(N841I) 4.1
nM
AC220 FLT3(D835H) 3.7
nM
AC220 KIT(A829P) 3.6
nM