AC220 KINOMEscan - Dataset (ID:20147)

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Small Molecule Protein Kd Conc unit
AC220 KIT 4.8
nM
AC220 KIT(A829P) 3.6
nM
AC220 KIT(D816H) 320.0
nM
AC220 KIT(D816V) 150.0
nM
AC220 KIT(L576P) 6.3
nM
AC220 KIT(V559D) 5.0
nM
AC220 KIT(V559D,T670I) 6.0
nM
AC220 KIT(V559D,V654A) 36.0
nM
AC220 LATS1
nM
AC220 LATS2
nM
AC220 LCK 2500.0
nM
AC220 LIMK1
nM
AC220 LIMK2
nM
AC220 LKB1
nM
AC220 LOK 2100.0
nM
AC220 LRRK2
nM
AC220 LRRK2(G2019S)
nM
AC220 LTK
nM
AC220 LYN 5700.0
nM
AC220 M3K13
nM
AC220 MAK
nM
AC220 MAP3K1
nM
AC220 MAP3K15
nM
AC220 M3K2
nM
AC220 MAP3K3
nM