AC220 KINOMEscan - Dataset (ID:20147)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
AC220 | KIT | 4.8 | nM |
AC220 | KIT(A829P) | 3.6 | nM |
AC220 | KIT(D816H) | 320.0 | nM |
AC220 | KIT(D816V) | 150.0 | nM |
AC220 | KIT(L576P) | 6.3 | nM |
AC220 | KIT(V559D) | 5.0 | nM |
AC220 | KIT(V559D,T670I) | 6.0 | nM |
AC220 | KIT(V559D,V654A) | 36.0 | nM |
AC220 | LATS1 | nM | |
AC220 | LATS2 | nM | |
AC220 | LCK | 2500.0 | nM |
AC220 | LIMK1 | nM | |
AC220 | LIMK2 | nM | |
AC220 | LKB1 | nM | |
AC220 | LOK | 2100.0 | nM |
AC220 | LRRK2 | nM | |
AC220 | LRRK2(G2019S) | nM | |
AC220 | LTK | nM | |
AC220 | LYN | 5700.0 | nM |
AC220 | M3K13 | nM | |
AC220 | MAK | nM | |
AC220 | MAP3K1 | nM | |
AC220 | MAP3K15 | nM | |
AC220 | M3K2 | nM | |
AC220 | MAP3K3 | nM |