Dabrafenib KINOMEscan - Dataset (ID:20131)

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Small Molecule Protein % Control Assay compound conc Conc unit
Dabrafenib ABL1(F317L)-phosphorylated 48.0 10
uM
Dabrafenib ABL1(F317L)-nonphosphorylated 14.0 10
uM
Dabrafenib ABL1(F317I)-phosphorylated 59.0 10
uM
Dabrafenib ABL1(F317I)-nonphosphorylated 30.0 10
uM
Dabrafenib ABL1(E255K)-phosphorylated 14.0 10
uM
Dabrafenib AAK1 26.0 10
uM