Dabrafenib KINOMEscan - Dataset (ID:20131)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200077 CDK4-cyclinD1 200077 P11802
Cyclin-dependent kinase 4; cell division protein kinase 4
KINOMEscan Wild Type; Full length
200062 CAMK1G 200062 Q96NX5
Calcium/calmodulin-dependent protein kinase IG; CAMK1G; CLICKIII; dJ272L16.1; VWS1
KINOMEscan Wild Type; Partial length
200063 CAMK2A 200063 Q9UQM7
Calcium/calmodulin-dependent protein kinase II alpha; CAMK2A; CAMKA; KIAA0968
KINOMEscan Wild Type; Partial length
200064 CAMK2B 200064 Q13554
Calcium/calmodulin-dependent protein kinase II beta; CAM2; CAMK2; CAMK2B; CAMKB; MGC29528
KINOMEscan Wild Type; Partial length
200043 M3K6 200043 O95382
Mitogen-activated protein kinase kinase kinase 6; ASK2; MAP3K6; MAPKKK6; MEKK6; MEKK6/MAP3K6; MGC125653; MGC20114
KINOMEscan Wild Type; Partial length
200066 CAMK2G 200066 Q13555
Calcium/calmodulin-dependent protein kinase II gamma; CAMK; CAMK2G; CAMKG; CAMK-II; FLJ16043; MGC26678
KINOMEscan Wild Type; Partial length
200075 CDK2 200075 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KINOMEscan Wild Type; Full length
200068 KKCC1 200068 Q8N5S9
Calcium/calmodulin-dependent protein kinase kinase 1, CaM-kinase IV kinase; CAMKK1; CAMKKA; DKFZp761M0423; MGC34095
KINOMEscan Wild Type; Partial length
200074 CDK11 200074 Q9BWU1
Cyclin-dependent kinase 19; bA346C16.3; CDC2L6; CDK11; CDK19; KIAA1028
KINOMEscan Wild Type; Partial length
200070 CASK 200070 O14936
Calcium/calmodulin-dependent serine protein kinase (MAGUK family); CAGH39; CAMGUK; CASK; CMG; FGS4; FLJ22219; FLJ31914; LIN2; MICPCH; TNRC8
KINOMEscan Wild Type; Partial length
200071 CDC2L1 200071 P21127
Cyclin-dependent kinase 11B; CDC2L1; CDC2L2; CDK11; CDK11B; CDK11-p110; CDK11-p46; CDK11-p58; CLK-1; FLJ59152; p58; p58CDC2L1; p58CLK-1; PITSLRE; PK58
KINOMEscan Wild Type; Partial length
200072 CDC2L2 200072 Q9UQ88
Cyclin-dependent kinase 11A; CDC2L2; CDC2L3; CDK11A; CDK11-p110; CDK11-p46; CDK11-p58; MGC131975; p58GTA; PITSLRE
KINOMEscan Wild Type; Partial length
200073 CDC2L5 200073 Q14004
Cyclin-dependent kinase 13; CDC2L; CDC2L5; CDK13; CHED; FLJ35215; KIAA1791
KINOMEscan Wild Type; Partial length
200042 M3K5 200042 Q99683
Mitogen-activated protein kinase kinase kinase 5; ASK; ASK/MAP3K5; ASK1; MAP3K5; MAPKKK5; MEKK5
KINOMEscan Wild Type; Partial length
200041 NUAK1 200041 O60285
NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1
KINOMEscan Wild Type; Partial length
200076 CDK3 200076 Q00526
Cyclin-dependent kinase 3; CDK3
KINOMEscan Wild Type; Full length
200027 ACVR1 200027 Q04771
Activin A receptor, type I; ACTRI; ACVR1; ACVR1A; ACVRLK2; ALK2; FOP; SKR1; TSRI
KINOMEscan Wild Type; Partial length
200078 CDK4-cyclinD3 200078 P11802
Cyclin-dependent kinase 4; cell division protein kinase 4
KINOMEscan Wild Type; Full length
200079 CDK5 200079 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KINOMEscan Wild Type; Full length
200080 CDK7 200080 P50613
Cyclin-dependent kinase 7; cell division protein kinase 7; CAK1; CDK7; CDKN7; MO15; p39MO15; STK1
KINOMEscan Wild Type; Full length
200026 ABL2 200026 P42684
V-abl Abelson murine leukemia viral oncogene homolog 2 (arg, Abelson-related gene); ABL2; ABLL; ARG; FLJ22224; FLJ31718; FLJ41441
KINOMEscan Wild Type; Partial length
200082 CDK9 200082 P50750
Cyclin-dependent kinase 9; cell division protein kinase 9; C-2k; CDC2L4; CDK9; CTK1; PITALRE; TAK
KINOMEscan Wild Type; Full length
200083 CDKL1 200083 Q00532
Cyclin-dependent kinase-like 1 (CDC2-related kinase); CDKL1; KKIALRE; P42
KINOMEscan Wild Type; Full length
200084 CDKL2 200084 Q92772
Cyclin-dependent kinase-like 2 (CDC2-related kinase); CDKL2; KKIAMRE; P56
KINOMEscan Wild Type; Partial length
200001 AAK1 200001 Q2M2I8
AP2 associated kinase 1; AAK1; DKFZp686F03202; DKFZp686K16132; FLJ23712; FLJ25931; FLJ31060; FLJ42882; FLJ45252; KIAA1048; MGC138170; MGC164568; MGC164570
KINOMEscan Wild Type; Partial length