Dabrafenib KINOMEscan - Dataset (ID:20131)
Proteins Studied
Download: Excel (XLSX), Comma-separated (CSV)
LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200468 | MLTK | 200468 | Q9NYL2 | Mitogen-activated protein kinase kinase kinase MLT; sterile alpha motif and leucine zipper containing kinase AZK; AZK; MLK7; mlklak; MLT; MLTK; MRK; pk; ZAK | KINOMEscan | Wild Type; Partial length | |||
200469 | ZAP70 | 200469 | P43403 | Tyrosine-protein kinase ZAP-70; Zeta-chain (TCR) associated protein kinase 70kDa; FLJ17670; FLJ17679; SRK; STD; TZK; ZAP70; ZAP-70 | KINOMEscan | Wild Type; Partial length | |||
200470 | BUB1 | 200470 | Budding uninhibited by benzimidazoles 1 homolog (yeast); BUB1A; BUB1L; hBUB1 | KINOMEscan | |||||
200471 | CSF1R-autoinhibited | 200471 | P07333 | Colony stimulating factor 1 receptor; CD115; C-FMS; CSF1R; CSF-1R; CSF-1-R; CSFR; FIM2; FIM-2; FMS; Fms/CSFR | KINOMEscan | ||||
200472 | FLT3-autoinhibited | 200472 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ||||
200473 | HASP | 200473 | Q8TF76 | Serine/threonine-protein kinase haspin; germ cell associated 2 (haspin); GSG2; HASPIN | KINOMEscan | ||||
200474 | KIT-autoinhibited | 200474 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | ||||
200475 | RSK2(Kin.Dom.2-C-terminal) | 200475 | P51812 | Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2 | KINOMEscan | Kin.Dom.2-C-terminal | |||
200476 | SGK1 | 200476 | O00141 | Serine/threonine-protein kinase Sgk1; serum/glucocorticoid regulated kinase 1; SGK | KINOMEscan | ||||
200477 | WNK1 | 200477 | Q9H4A3 | WNK lysine deficient protein kinase 1; KDP; PSK; p65; HSN2; HSAN2; PRKWNK1 | KINOMEscan | ||||
200478 | WNK3 | 200478 | Q9BYP7 | WNK lysine deficient protein kinase 3; PRKWNK3 | KINOMEscan | ||||
200479 | ALK(C1156Y) | 200479 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | C1156Y | |||
200480 | ALK(L1196M) | 200480 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | L1196M | |||
200481 | NEK10 | 200481 | Q6ZWH5 | NIMA (never in mitosis gene a)- related kinase 10 | KINOMEscan | ||||
201107 | MAP3K14 | 201107 | Q99558 | Mitogen-activated protein kinase kinase kinase 14; NF-kappa-beta-inducing kinase; NIK | KINOMEscan | ||||
200001 | AAK1 | 200001 | Q2M2I8 | AP2 associated kinase 1; AAK1; DKFZp686F03202; DKFZp686K16132; FLJ23712; FLJ25931; FLJ31060; FLJ42882; FLJ45252; KIAA1048; MGC138170; MGC164568; MGC164570 | KINOMEscan | Wild Type; Partial length | |||
201108 | SGK2 | 201108 | Q9HBY8 | Serine/threonine-protein kinase Sgk2; Serum/glucocorticoid-regulated kinase 2 | KINOMEscan | ||||
200026 | ABL2 | 200026 | P42684 | V-abl Abelson murine leukemia viral oncogene homolog 2 (arg, Abelson-related gene); ABL2; ABLL; ARG; FLJ22224; FLJ31718; FLJ41441 | KINOMEscan | Wild Type; Partial length | |||
200027 | ACVR1 | 200027 | Q04771 | Activin A receptor, type I; ACTRI; ACVR1; ACVR1A; ACVRLK2; ALK2; FOP; SKR1; TSRI | KINOMEscan | Wild Type; Partial length | |||
200028 | ACVR1B | 200028 | P36896 | Activin A receptor, type IB; ACTRIB; ACVR1B; ACVRLK4; ALK4; SKR2 | KINOMEscan | Wild Type; Partial length | |||
200029 | ACVR2A | 200029 | P27037 | Activin A receptor, type IIA; ActR2; ACTRII; ACVR2; ACVR2A | KINOMEscan | Wild Type; Partial length | |||
200030 | ACVR2B | 200030 | Q13705 | Activin A receptor, type IIB; ActR2B; ACTRIIB; ActR-IIB; ACVR2B; MGC116908 | KINOMEscan | Wild Type; Partial length | |||
200031 | ACVRL1 | 200031 | P37023 | Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I | KINOMEscan | Wild Type; Partial length | |||
200032 | ADCK3 | 200032 | Q8NI60 | Chaperone, ABC1 activity of bc1 complex homolog (S. pombe); ADCK3; ARCA2; CABC1; COQ8; MGC4849; SCAR9 | KINOMEscan | Wild Type; Full length | |||
200033 | ADCK4 | 200033 | Q96D53 | AarF domain containing kinase 4; ADCK4; FLJ12229 | KINOMEscan | Wild Type; Full length |