(R)-Roscovitine KINOMEscan - Dataset (ID:20124)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200220 KIT(V559D,T670I) 200220 P10721
V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR
KINOMEscan V559D,T670I Mutation (V559D,T670I); Partial length
200221 KIT(V559D,V654A) 200221 P10721
V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR
KINOMEscan V559D,V654A Mutation (V559D,V654A); Partial length
200055 BRAF(V600E) 200055 P15056
V-raf murine sarcoma viral oncogene homolog B1; BRAF; BRAF1; B-RAF1; FLJ95109; MGC126806; MGC138284; RAFB1
KINOMEscan V600E Mutation (V600E); Partial length
200372 RET(V804L) 200372 P07949
Proto-oncogene tyrosine-protein kinase receptor Ret; CDHF12; CDHR16; HSCR1; MEN2A; MEN2B; MTC1; PTC; RET; RET51; RET-ELE1
KINOMEscan V804L Mutation (V804L); Partial length
200373 RET(V804M) 200373 P07949
Proto-oncogene tyrosine-protein kinase receptor Ret; CDHF12; CDHR16; HSCR1; MEN2A; MEN2B; MTC1; PTC; RET; RET51; RET-ELE1
KINOMEscan V804M Mutation (V804M); Partial length
200261 MET(Y1235D) 200261 P08581
Hepatocyte growth factor receptor; AUTS9; c-Met; HGFR; MET; RCCP2
KINOMEscan Y1235D Mutation (Y1235D); Partial length
200023 ABL1(Y253F)-phosphorylated 200023 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan Y253F phosphorylated Mutation (Y253F); Partial length
200071 CDC2L1 200071 P21127
Cyclin-dependent kinase 11B; CDC2L1; CDC2L2; CDK11; CDK11B; CDK11-p110; CDK11-p46; CDK11-p58; CLK-1; FLJ59152; p58; p58CDC2L1; p58CLK-1; PITSLRE; PK58
KINOMEscan Wild Type; Partial length
200040 ANKK1 200040 Q8NFD2
Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288
KINOMEscan Wild Type; Partial length
200070 CASK 200070 O14936
Calcium/calmodulin-dependent serine protein kinase (MAGUK family); CAGH39; CAMGUK; CASK; CMG; FGS4; FLJ22219; FLJ31914; LIN2; MICPCH; TNRC8
KINOMEscan Wild Type; Partial length
200069 CAMKK2 200069 Q96RR4
Calcium/calmodulin-dependent protein kinase kinase 2, beta; CAMKK; CAMKK2; CAMKKB; KIAA0787; MGC15254
KINOMEscan Wild Type; Partial length
200072 CDC2L2 200072 Q9UQ88
Cyclin-dependent kinase 11A; CDC2L2; CDC2L3; CDK11A; CDK11-p110; CDK11-p46; CDK11-p58; MGC131975; p58GTA; PITSLRE
KINOMEscan Wild Type; Partial length
200039 AMPK-alpha2 200039 P54646
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2
KINOMEscan Wild Type; Partial length
200068 KKCC1 200068 Q8N5S9
Calcium/calmodulin-dependent protein kinase kinase 1, CaM-kinase IV kinase; CAMKK1; CAMKKA; DKFZp761M0423; MGC34095
KINOMEscan Wild Type; Partial length
200067 KCC4 200067 Q16566
Calcium/calmodulin-dependent protein kinase type IV; CAMK4; CaMK-GR; MGC36771
KINOMEscan Wild Type; Partial length
200066 CAMK2G 200066 Q13555
Calcium/calmodulin-dependent protein kinase II gamma; CAMK; CAMK2G; CAMKG; CAMK-II; FLJ16043; MGC26678
KINOMEscan Wild Type; Partial length
200065 KCC2D 200065 Q13557
Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911
KINOMEscan Wild Type; Partial length
200038 AMPK-alpha1 200038 Q13131
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1
KINOMEscan Wild Type; Partial length
200037 ALK 200037 Q9UM73
Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK
KINOMEscan Wild Type; Partial length
200064 CAMK2B 200064 Q13554
Calcium/calmodulin-dependent protein kinase II beta; CAM2; CAMK2; CAMK2B; CAMKB; MGC29528
KINOMEscan Wild Type; Partial length
200063 CAMK2A 200063 Q9UQM7
Calcium/calmodulin-dependent protein kinase II alpha; CAMK2A; CAMKA; KIAA0968
KINOMEscan Wild Type; Partial length
200036 AKT3 200036 Q9Y243
V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2
KINOMEscan Wild Type; Partial length
200062 CAMK1G 200062 Q96NX5
Calcium/calmodulin-dependent protein kinase IG; CAMK1G; CLICKIII; dJ272L16.1; VWS1
KINOMEscan Wild Type; Partial length
200061 CAMK1D 200061 Q8IU85
Calcium/calmodulin-dependent protein kinase ID; CaM-K1; CAMK1D; CaMKID; CKLiK
KINOMEscan Wild Type; Partial length
200035 AKT2 200035 P31751
V-akt murine thymoma viral oncogene homolog 2; AKT2; Akt2/PKBb; PKBb; PKBBETA; PRKBB; RAC-BETA
KINOMEscan Wild Type; Partial length