XMD-12 KINOMEscan - Dataset (ID:20115)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
XMD-12 | ABL1(M351T)-phosphorylated | 3.0 | 1 | uM |
XMD-12 | ABL1-nonphosphorylated | 3.2 | 1 | uM |
XMD-12 | ABL1(F317L)-phosphorylated | 3.3 | 1 | uM |
XMD-12 | ABL1(T315I)-nonphosphorylated | 3.6 | 1 | uM |
XMD-12 | ABL1-phosphorylated | 3.6 | 1 | uM |
XMD-12 | RET(M918T) | 4.2 | 1 | uM |
XMD-12 | PIK3CG | 4.2 | 1 | uM |
XMD-12 | JAK1(JH2domain-pseudokinase) | 4.8 | 1 | uM |
XMD-12 | SgK110 | 5.4 | 1 | uM |
XMD-12 | CSF1R | 5.8 | 1 | uM |
XMD-12 | ULK2 | 6.2 | 1 | uM |
XMD-12 | FGR | 6.6 | 1 | uM |
XMD-12 | ABL1(F317I)-phosphorylated | 7.4 | 1 | uM |
XMD-12 | MKNK2 | 8.4 | 1 | uM |
XMD-12 | BLK | 12.0 | 1 | uM |
XMD-12 | BMPR1B | 13.0 | 1 | uM |
XMD-12 | RET | 15.0 | 1 | uM |
XMD-12 | ULK1 | 16.0 | 1 | uM |
XMD-12 | AMPK-alpha1 | 17.0 | 1 | uM |
XMD-12 | NUAK1 | 17.0 | 1 | uM |
XMD-12 | ABL1(F317L)-nonphosphorylated | 20.0 | 1 | uM |
XMD-12 | SRC | 21.0 | 1 | uM |
XMD-12 | AURKC | 22.0 | 1 | uM |
XMD-12 | SNARK | 23.0 | 1 | uM |
XMD-12 | FLT3(D835Y) | 24.0 | 1 | uM |