XMD-12 KINOMEscan - Dataset (ID:20115)

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Small Molecule Protein % Control Assay compound conc Conc unit
XMD-12 ABL1(M351T)-phosphorylated 3.0 1
uM
XMD-12 ABL1-nonphosphorylated 3.2 1
uM
XMD-12 ABL1(F317L)-phosphorylated 3.3 1
uM
XMD-12 ABL1(T315I)-nonphosphorylated 3.6 1
uM
XMD-12 ABL1-phosphorylated 3.6 1
uM
XMD-12 RET(M918T) 4.2 1
uM
XMD-12 PIK3CG 4.2 1
uM
XMD-12 JAK1(JH2domain-pseudokinase) 4.8 1
uM
XMD-12 SgK110 5.4 1
uM
XMD-12 CSF1R 5.8 1
uM
XMD-12 ULK2 6.2 1
uM
XMD-12 FGR 6.6 1
uM
XMD-12 ABL1(F317I)-phosphorylated 7.4 1
uM
XMD-12 MKNK2 8.4 1
uM
XMD-12 BLK 12.0 1
uM
XMD-12 BMPR1B 13.0 1
uM
XMD-12 RET 15.0 1
uM
XMD-12 ULK1 16.0 1
uM
XMD-12 AMPK-alpha1 17.0 1
uM
XMD-12 NUAK1 17.0 1
uM
XMD-12 ABL1(F317L)-nonphosphorylated 20.0 1
uM
XMD-12 SRC 21.0 1
uM
XMD-12 AURKC 22.0 1
uM
XMD-12 SNARK 23.0 1
uM
XMD-12 FLT3(D835Y) 24.0 1
uM