XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 7.1 | 10 | uM |
XMD-12 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -71.5 | 10 | uM |
XMD-12 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 72.5 | 10 | uM |
XMD-12 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.3 | 10 | uM |
XMD-12 | PC-3 | PDK1 | EYAIkILEK | Lys1 | -7.3 | 10 | uM |
XMD-12 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 73.5 | 10 | uM |
XMD-12 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -7.5 | 10 | uM |
XMD-12 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -7.5 | 10 | uM |
XMD-12 | PC-3 | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -7.5 | 10 | uM |
XMD-12 | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 75.4 | 10 | uM |
XMD-12 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 75.9 | 10 | uM |
XMD-12 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -7.6 | 10 | uM |
XMD-12 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 76.2 | 10 | uM |
XMD-12 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -8.0 | 10 | uM |
XMD-12 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 81.1 | 10 | uM |
XMD-12 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 81.3 | 10 | uM |
XMD-12 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 8.2 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | 8.4 | 10 | uM |
XMD-12 | PC-3 | LOK | NKETGALAAAkVIETK | Lys1 | 84.5 | 10 | uM |
XMD-12 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.5 | 10 | uM |
XMD-12 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 85.4 | 10 | uM |
XMD-12 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | -8.6 | 10 | uM |
XMD-12 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 87.9 | 10 | uM |
XMD-12 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |
XMD-12 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 88.7 | 10 | uM |