XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
7.1
10
uM
XMD-12 HeLa MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-71.5
10
uM
XMD-12 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
72.5
10
uM
XMD-12 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-7.3
10
uM
XMD-12 PC-3 PDK1
EYAIkILEK
Lys1
-7.3
10
uM
XMD-12 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
73.5
10
uM
XMD-12 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-7.5
10
uM
XMD-12 HeLa NEK9
DIkTLNIFLTK
Lys2
-7.5
10
uM
XMD-12 PC-3 MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-7.5
10
uM
XMD-12 PC-3 M3K2
ELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
75.4
10
uM
XMD-12 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
75.9
10
uM
XMD-12 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-7.6
10
uM
XMD-12 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
76.2
10
uM
XMD-12 HeLa KS6B2
DLkPENIMLSSQGHIK
Lys2
-8.0
10
uM
XMD-12 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
81.1
10
uM
XMD-12 PC-3 CDK10
DLkVSNLLMTDK
Lys2
81.3
10
uM
XMD-12 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
8.2
10
uM
XMD-12 PC-3 EPHA2
EVPVAIkTLK
Lys1
8.4
10
uM
XMD-12 PC-3 LOK
NKETGALAAAkVIETK
Lys1
84.5
10
uM
XMD-12 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
-8.5
10
uM
XMD-12 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
85.4
10
uM
XMD-12 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
-8.6
10
uM
XMD-12 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
87.9
10
uM
XMD-12 HeLa SGK3
FYAVkVLQK
Lys1
-8.8
10
uM
XMD-12 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
88.7
10
uM