XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -16.3 | 10 | uM |
XMD-12 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | -16.3 | 10 | uM |
XMD-12 | PC-3 | PKCa,PKCb | DLkLDNVMLDSEGHIK | Lys2 | 16.5 | 10 | uM |
XMD-12 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -16.7 | 10 | uM |
XMD-12 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -16.8 | 10 | uM |
XMD-12 | PC-3 | ATR | FYIMMCkPK | ATP | 16.8 | 10 | uM |
XMD-12 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -17.2 | 10 | uM |
XMD-12 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -17.4 | 10 | uM |
XMD-12 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 17.6 | 10 | uM |
XMD-12 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | 1.8 | 10 | uM |
XMD-12 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 18.0 | 10 | uM |
XMD-12 | HeLa | PKD1,PKD2 | NIVHCDLkPENVLLASADPFPQVK | Lys2 | 18.2 | 10 | uM |
XMD-12 | HeLa | RIPK3 | DLkPSNVLLDPELHVK | Lys2 | 1.9 | 10 | uM |
XMD-12 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 1.9 | 10 | uM |
XMD-12 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.3 | 10 | uM |
XMD-12 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -19.8 | 10 | uM |
XMD-12 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -20.0 | 10 | uM |
XMD-12 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 20.0 | 10 | uM |
XMD-12 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -20.1 | 10 | uM |
XMD-12 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -20.4 | 10 | uM |
XMD-12 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | -20.6 | 10 | uM |
XMD-12 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -208.2 | 10 | uM |
XMD-12 | HeLa | ATR | FYIMMCkPK | ATP | -2.1 | 10 | uM |
XMD-12 | HeLa | SYK | ISDFGLSkALR | Activation Loop | 2.1 | 10 | uM |
XMD-12 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -21.4 | 10 | uM |