XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-16.3
10
uM
XMD-12 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
-16.3
10
uM
XMD-12 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
16.5
10
uM
XMD-12 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-16.7
10
uM
XMD-12 HeLa CaMK1a
LVAIkCIAK
Lys1
-16.8
10
uM
XMD-12 PC-3 ATR
FYIMMCkPK
ATP
16.8
10
uM
XMD-12 HeLa NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-17.2
10
uM
XMD-12 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
-17.4
10
uM
XMD-12 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
17.6
10
uM
XMD-12 HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
1.8
10
uM
XMD-12 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
18.0
10
uM
XMD-12 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
18.2
10
uM
XMD-12 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
1.9
10
uM
XMD-12 PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
1.9
10
uM
XMD-12 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
19.3
10
uM
XMD-12 HeLa JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-19.8
10
uM
XMD-12 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-20.0
10
uM
XMD-12 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
20.0
10
uM
XMD-12 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-20.1
10
uM
XMD-12 HeLa p38a
DLkPSNLAVNEDCELK
Lys2
-20.4
10
uM
XMD-12 HeLa PKN1
GHFGkVLLSEFRPSGELFAIK
Lys1
-20.6
10
uM
XMD-12 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-208.2
10
uM
XMD-12 HeLa ATR
FYIMMCkPK
ATP
-2.1
10
uM
XMD-12 HeLa SYK
ISDFGLSkALR
Activation Loop
2.1
10
uM
XMD-12 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-21.4
10
uM