XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 12.5 | 10 | uM |
| XMD-12 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -12.6 | 10 | uM |
| XMD-12 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -12.6 | 10 | uM |
| XMD-12 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | 12.8 | 10 | uM |
| XMD-12 | HeLa | MYO3A,MYO3B | DVkGNNILLTTEGGVK | Lys2 | -1.3 | 10 | uM |
| XMD-12 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | -13.0 | 10 | uM |
| XMD-12 | HeLa | PAN3 | VMDPTkILITGK | -13.7 | 10 | uM | |
| XMD-12 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -13.9 | 10 | uM |
| XMD-12 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 14.0 | 10 | uM |
| XMD-12 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -14.1 | 10 | uM |
| XMD-12 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 14.3 | 10 | uM |
| XMD-12 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 14.4 | 10 | uM |
| XMD-12 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 14.6 | 10 | uM |
| XMD-12 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 14.8 | 10 | uM |
| XMD-12 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | 14.9 | 10 | uM |
| XMD-12 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -1.5 | 10 | uM |
| XMD-12 | PC-3 | SNRK | DLkPENVVFFEK | Lys2 | -15.0 | 10 | uM |
| XMD-12 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 15.0 | 10 | uM |
| XMD-12 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 15.0 | 10 | uM |
| XMD-12 | PC-3 | MAP2K4 | MVHKPSGQIMAVkR | Lys1 | 15.1 | 10 | uM |
| XMD-12 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 15.2 | 10 | uM |
| XMD-12 | PC-3 | RON | IQCAIkSLSR | Lys1 | 15.8 | 10 | uM |
| XMD-12 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 15.8 | 10 | uM |
| XMD-12 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -1.6 | 10 | uM |
| XMD-12 | PC-3 | MAP2K3 | DVkPSNVLINK | Lys2 | 1.6 | 10 | uM |