XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD-12 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 24.9 | 10 | uM |
| XMD-12 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 64.7 | 10 | uM |
| XMD-12 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -4.5 | 10 | uM |
| XMD-12 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.5 | 10 | uM |
| XMD-12 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 2.9 | 10 | uM |
| XMD-12 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -16.7 | 10 | uM |
| XMD-12 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -9.6 | 10 | uM |
| XMD-12 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -17.4 | 10 | uM |
| XMD-12 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -10.0 | 10 | uM |
| XMD-12 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | 3.4 | 10 | uM |
| XMD-12 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -7.5 | 10 | uM |
| XMD-12 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | -26.4 | 10 | uM |
| XMD-12 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | 69.0 | 10 | uM |
| XMD-12 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 72.5 | 10 | uM |
| XMD-12 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 38.2 | 10 | uM |
| XMD-12 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | -4.1 | 10 | uM |
| XMD-12 | HeLa | SLK | DLkAGNILFTLDGDIK | Lys2 | 6.8 | 10 | uM |
| XMD-12 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 42.0 | 10 | uM |
| XMD-12 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 40.3 | 10 | uM |
| XMD-12 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 2.8 | 10 | uM |
| XMD-12 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | -10.1 | 10 | uM |
| XMD-12 | PC-3 | PKCa,PKCb | DLkLDNVMLDSEGHIK | Lys2 | 16.5 | 10 | uM |
| XMD-12 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 10.9 | 10 | uM |
| XMD-12 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -4.3 | 10 | uM |
| XMD-12 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 7.1 | 10 | uM |