XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
88.8
10
uM
XMD-12 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
90.3
10
uM
XMD-12 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
91.3
10
uM
XMD-12 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
91.5
10
uM
XMD-12 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.2
10
uM
XMD-12 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
92.9
10
uM
XMD-12 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-9.3
10
uM
XMD-12 HeLa MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
93.5
10
uM
XMD-12 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
94.6
10
uM
XMD-12 HeLa PKR
DLkPSNIFLVDTK
Lys2
-9.5
10
uM
XMD-12 HeLa AurB
SHFIVALkVLFK
Lys1
95.0
10
uM
XMD-12 PC-3 MAP2K4
DIkPSNILLDR
Lys2
-9.6
10
uM
XMD-12 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
97.4
10
uM
XMD-12 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
10
uM
XMD-12 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD-12 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
10
uM