XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
75.9
10
uM
XMD-12 PC-3 AGK
ATVFLNPAACkGK
ATP
-6.7
10
uM
XMD-12 HeLa PIK3CG
KkPLWLEFK
ATP
5.4
10
uM
XMD-12 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
30.5
10
uM
XMD-12 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
51.4
10
uM
XMD-12 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
-5.5
10
uM
XMD-12 PC-3 ATR
FYIMMCkPK
ATP
16.8
10
uM
XMD-12 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
5.9
10
uM
XMD-12 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
60.5
10
uM
XMD-12 HeLa PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
23.7
10
uM
XMD-12 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
26.6
10
uM
XMD-12 HeLa ATR
FYIMMCkPK
ATP
-2.1
10
uM
XMD-12 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
76.2
10
uM
XMD-12 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-25.3
10
uM
XMD-12 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
33.9
10
uM
XMD-12 HeLa PI4KB
VPHTQAVVLNSkDK
ATP
-5.8
10
uM
XMD-12 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
0.2
10
uM
XMD-12 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
-11.2
10
uM
XMD-12 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
-11.6
10
uM
XMD-12 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-1.6
10
uM
XMD-12 HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
-6.2
10
uM
XMD-12 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
14.4
10
uM
XMD-12 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
-16.3
10
uM
XMD-12 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
22.4
10
uM
XMD-12 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
33.0
10
uM