XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 75.9 | 10 | uM |
XMD-12 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -6.7 | 10 | uM |
XMD-12 | HeLa | PIK3CG | KkPLWLEFK | ATP | 5.4 | 10 | uM |
XMD-12 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 30.5 | 10 | uM |
XMD-12 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 51.4 | 10 | uM |
XMD-12 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | -5.5 | 10 | uM |
XMD-12 | PC-3 | ATR | FYIMMCkPK | ATP | 16.8 | 10 | uM |
XMD-12 | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | 5.9 | 10 | uM |
XMD-12 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 60.5 | 10 | uM |
XMD-12 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 23.7 | 10 | uM |
XMD-12 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 26.6 | 10 | uM |
XMD-12 | HeLa | ATR | FYIMMCkPK | ATP | -2.1 | 10 | uM |
XMD-12 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 76.2 | 10 | uM |
XMD-12 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -25.3 | 10 | uM |
XMD-12 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 33.9 | 10 | uM |
XMD-12 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -5.8 | 10 | uM |
XMD-12 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.2 | 10 | uM |
XMD-12 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | -11.2 | 10 | uM |
XMD-12 | HeLa | PRPK | FLSGLELVkQGAEAR | ATP Loop | -11.6 | 10 | uM |
XMD-12 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -1.6 | 10 | uM |
XMD-12 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | -6.2 | 10 | uM |
XMD-12 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | 14.4 | 10 | uM |
XMD-12 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | -16.3 | 10 | uM |
XMD-12 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 22.4 | 10 | uM |
XMD-12 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 33.0 | 10 | uM |