XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-14.1
 10
uM
XMD-12 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-23.4
 10
uM
XMD-12 HeLa DMPK
DIkPDNILLDR
Lys2
-4.3
 10
uM
XMD-12 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
75.9
 10
uM
XMD-12 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
30.5
 10
uM
XMD-12 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
51.4
 10
uM
XMD-12 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.2
 10
uM
XMD-12 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-2.6
 10
uM
XMD-12 PC-3 EGFR
IPVAIkELR
Lys1
-0.3
 10
uM
XMD-12 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
2.2
 10
uM
XMD-12 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-16.3
 10
uM
XMD-12 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
-24.1
 10
uM
XMD-12 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
97.4
 10
uM
XMD-12 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
85.4
 10
uM
XMD-12 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
30.6
 10
uM
XMD-12 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
42.4
 10
uM
XMD-12 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
70.5
 10
uM
XMD-12 HeLa GCK
DTVTSELAAVkIVK
Lys1
15.0
 10
uM
XMD-12 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
0.2
 10
uM
XMD-12 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-16.7
 10
uM
XMD-12 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
2.9
 10
uM
XMD-12 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-7.3
 10
uM
XMD-12 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
24.9
 10
uM
XMD-12 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
64.7
 10
uM
XMD-12 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
-11.9
 10
uM