XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD16-144 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -2.0 | 10 | uM |
XMD16-144 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 13.9 | 10 | uM |
XMD16-144 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -6.6 | 10 | uM |
XMD16-144 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 82.5 | 10 | uM |
XMD16-144 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 46.1 | 10 | uM |
XMD16-144 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 73.5 | 10 | uM |
XMD16-144 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 0.2 | 10 | uM |
XMD16-144 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -3.6 | 10 | uM |
XMD16-144 | PC-3 | EGFR | IPVAIkELR | Lys1 | 3.7 | 10 | uM |
XMD16-144 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 4.4 | 10 | uM |
XMD16-144 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -11.9 | 10 | uM |
XMD16-144 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 14.5 | 10 | uM |
XMD16-144 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.5 | 10 | uM |
XMD16-144 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 80.3 | 10 | uM |
XMD16-144 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 28.5 | 10 | uM |
XMD16-144 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 51.1 | 10 | uM |
XMD16-144 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 66.9 | 10 | uM |
XMD16-144 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 3.1 | 10 | uM |
XMD16-144 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | -4.6 | 10 | uM |
XMD16-144 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -3.2 | 10 | uM |
XMD16-144 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 27.7 | 10 | uM |
XMD16-144 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | 2.5 | 10 | uM |
XMD16-144 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -1.3 | 10 | uM |
XMD16-144 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 27.1 | 10 | uM |
XMD16-144 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 0.0 | 10 | uM |