XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa MLTK
WISQDKEVAVKk
Lys1
8.5
10
uM
XMD11-50 HeLa ILK
WQGNDIVVkVLK
Lys1
3.0
10
uM
XMD11-50 PC-3 ILK
WQGNDIVVkVLK
Lys1
16.3
10
uM
XMD11-50 HeLa TLK1
YAAVkIHQLNK
Lys1
8.2
10
uM
XMD11-50 PC-3 TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD11-50 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
11.2
10
uM
XMD11-50 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-17.5
10
uM
XMD11-50 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-18.4
10
uM
XMD11-50 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-5.3
10
uM
XMD11-50 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-0.8
10
uM
XMD11-50 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
8.2
10
uM
XMD11-50 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-10.3
10
uM
XMD11-50 PC-3 TLK2
YVAVkIHQLNK
Lys1
-0.3
10
uM
XMD11-50 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-9.2
10
uM