XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
13.2
10
uM
XMD11-50 PC-3 PI42C
ELPTLkDMDFLNK
ATP
29.2
10
uM
XMD11-50 PC-3 AGK
ATVFLNPAACkGK
ATP
5.8
10
uM
XMD11-50 HeLa PIK3CG
KkPLWLEFK
ATP
-10.0
10
uM
XMD11-50 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
6.5
10
uM
XMD11-50 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
11.9
10
uM
XMD11-50 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
14.1
10
uM
XMD11-50 PC-3 ATR
FYIMMCkPK
ATP
-10.3
10
uM
XMD11-50 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
25.2
10
uM
XMD11-50 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
14.3
10
uM
XMD11-50 HeLa ATR
FYIMMCkPK
ATP
2.5
10
uM
XMD11-50 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
53.0
10
uM
XMD11-50 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
41.8
10
uM
XMD11-50 HeLa PI4KB
VPHTQAVVLNSkDK
ATP
18.7
10
uM
XMD11-50 HeLa PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
6.5
10
uM
XMD11-50 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
12.4
10
uM
XMD11-50 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
-11.4
10
uM
XMD11-50 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-6.2
10
uM
XMD11-50 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
17.3
10
uM
XMD11-50 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
-1.1
10
uM
XMD11-50 HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
25.2
10
uM
XMD11-50 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
6.5
10
uM
XMD11-50 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
8.3
10
uM
XMD11-50 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
16.1
10
uM
XMD11-50 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
63.4
10
uM