Torin1 KiNativ -- single dose experiment - Dataset (ID:20094)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
Torin1 | HeLa | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 10.4 | 10 | uM |
Torin1 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -0.1 | 10 | uM |
Torin1 | HeLa | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -16.4 | 10 | uM |
Torin1 | HeLa | MAP2K3 | MCDFGISGYLVDSVAkTMDAGCKPYMAPER | Activation Loop | 13.0 | 10 | uM |
Torin1 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | 27.1 | 10 | uM |
Torin1 | HeLa | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 6.8 | 10 | uM |
Torin1 | HeLa | RSK1_domain1 | LTDFGLSkEAIDHEKK | Activation Loop | 5.0 | 10 | uM |
Torin1 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | 6.3 | 10 | uM |
Torin1 | HeLa | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 4.5 | 10 | uM |
Torin1 | HeLa | JAK1 domain2 | IGDFGLTkAIETDKEYYTVKDDR | Activation Loop | 38.2 | 10 | uM |
Torin1 | HeLa | MAP2K6 | MCDFGISGYLVDSVAkTIDAGCKPYMAPER | Activation Loop | 19.3 | 10 | uM |
Torin1 | HeLa | MST3,MST4,YSK1 | LADFGVAGQLTDTQIkR | Activation Loop | 8.6 | 10 | uM |
Torin1 | HeLa | NDR1,NDR2 | LSDFGLCTGLkK | Activation Loop | 13.2 | 10 | uM |
Torin1 | HeLa | PKR | IGDFGLVTSLkNDGKR | Activation Loop | -13.5 | 10 | uM |
Torin1 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -1.9 | 10 | uM |
Torin1 | HeLa | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | -1.9 | 10 | uM |
Torin1 | HeLa | FER | QEDGGVYSSSGLkQIPIKWTAPEALNYGR | Activation Loop | 2.2 | 10 | uM |
Torin1 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | -18.0 | 10 | uM |
Torin1 | HeLa | PIK3C3 | TEDGGkYPVIFKHGDDLR | ATP | 12.9 | 10 | uM |
Torin1 | HeLa | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | 14.5 | 10 | uM |
Torin1 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 14.2 | 10 | uM |
Torin1 | HeLa | FYV1 | GGkSGAAFYATEDDRFILK | ATP | 9.6 | 10 | uM |
Torin1 | HeLa | DNAPK | EHPFLVkGGEDLR | ATP | 76.2 | 10 | uM |
Torin1 | HeLa | DNAPK | GHDEREHPFLVkGGEDLR | ATP | 82.0 | 10 | uM |
Torin1 | HeLa | AGK | ATVFLNPAACkGK | ATP | -0.8 | 10 | uM |