Torin1 KiNativ -- single dose experiment - Dataset (ID:20094)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Torin1 HeLa SLK
AQNKETSVLAAAkVIDTK
Lys1
2.2
10
uM
Torin1 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
26.7
10
uM
Torin1 HeLa SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
18.7
10
uM
Torin1 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-3.5
10
uM
Torin1 HeLa TAOK2
DVkAGNILLSEPGLVK
Lys2
13.9
10
uM
Torin1 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
14.7
10
uM
Torin1 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
6.7
10
uM
Torin1 HeLa TLK2
YVAVkIHQLNK
Lys1
7.0
10
uM
Torin1 HeLa ULK3
EVVAIkCVAK
Lys1
5.4
10
uM
Torin1 HeLa ULK3
NISHLDLkPQNILLSSLEKPHLK
Lys2
21.5
10
uM
Torin1 HeLa VRK2
MLDVLEYIHENEYVHGDIkAANLLLGYK
Lys2
8.5
10
uM
Torin1 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
25.2
10
uM
Torin1 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-16.0
10
uM
Torin1 HeLa Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-16.4
10
uM
Torin1 HeLa YANK3
DVkPDNILLDER
Lys2
-0.5
10
uM
Torin1 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
6.9
10
uM