Torin1 KiNativ -- single dose experiment - Dataset (ID:20094)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Torin1 HeLa BRAF
SIIHRDLkSNNIFLHEDLTVKIGDFGLATVK
Lys2
-8.8
10
uM
Torin1 HeLa CDC2
RVLHRDLkPQNLLIDDK
Lys2
-33.5
10
uM
Torin1 HeLa CDK2
VLHRDLkPQNLLINTEGAIK
Lys2
24.1
10
uM
Torin1 HeLa CLK3
FLHENQLTHTDLkPENILFVNSEFETLYNEHK
Lys2
-9.2
10
uM
Torin1 HeLa LATS2
DIkPDNILIDLDGHIK
Lys2
1.1
10
uM
Torin1 HeLa PRP4
CNILHADIkPDNILVNESK
Lys2
3.8
10
uM
Torin1 HeLa RK
DLkPENVLLDNDGNVR
Lys2
13.2
10
uM
Torin1 HeLa CHK1
LSkGDGLEFK
Other
12.5
10
uM
Torin1 HeLa PRP4
AAGIGkDFKENPNLR
Other
2.5
10
uM
Torin1 HeLa ROCK1
kLQLELNQER
Other
-28.6
10
uM
Torin1 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
11.4
10
uM
Torin1 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Protein Kinase Domain
12.4
10
uM
Torin1 HeLa ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
4.5
10
uM
Torin1 HeLa MK14
QELNkTIWEVPER
Protein Kinase Domain
-9.8
10
uM
Torin1 HeLa ATR
kAGHHQTAYNALLNAGESR
Protein Kinase Domain
-4.0
10
uM
Torin1 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
17.1
10
uM