GSK1059615 KINOMEscan - Dataset (ID:20085)

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Small Molecule Protein % Control Assay compound conc Conc unit
GSK1059615 ABL1(F317L)-phosphorylated 60.0 10
uM
GSK1059615 ABL1(F317L)-nonphosphorylated 80.0 10
uM
GSK1059615 ABL1(F317I)-phosphorylated 79.0 10
uM
GSK1059615 ABL1(F317I)-nonphosphorylated 89.0 10
uM
GSK1059615 ABL1(E255K)-phosphorylated 71.0 10
uM
GSK1059615 AAK1 1.0 10
uM