GSK2126458 KINOMEscan - Dataset (ID:20084)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Omipalisib | ABL1(F317L)-phosphorylated | 70.0 | 10 | uM |
Omipalisib | ABL1(F317L)-nonphosphorylated | 71.0 | 10 | uM |
Omipalisib | ABL1(F317I)-phosphorylated | 64.0 | 10 | uM |
Omipalisib | ABL1(F317I)-nonphosphorylated | 100.0 | 10 | uM |
Omipalisib | ABL1(E255K)-phosphorylated | 54.0 | 10 | uM |
Omipalisib | AAK1 | 13.0 | 10 | uM |