WH-4-025 KINOMEscan - Dataset (ID:20056)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200221 KIT(V559D,V654A) 200221 P10721
V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR
KINOMEscan V559D,V654A Mutation (V559D,V654A); Partial length
200055 BRAF(V600E) 200055 P15056
V-raf murine sarcoma viral oncogene homolog B1; BRAF; BRAF1; B-RAF1; FLJ95109; MGC126806; MGC138284; RAFB1
KINOMEscan V600E Mutation (V600E); Partial length
200022 ABL1(Y253F) 200022 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan Y253F
200049 BLK 200049 P51451
Tyrosine-protein kinase BLK; B lymphoid tyrosine kinase; BLK; MGC10442
KINOMEscan Wild Type; Partial length
200048 BIKE 200048 Q9NSY1
BMP2 inducible kinase; BIKE; BMP2K; DKFZp434K0614; DKFZp434P0116; HRIHFB2017
KINOMEscan Wild Type; Partial length
200032 ADCK3 200032 Q8NI60
Chaperone, ABC1 activity of bc1 complex homolog (S. pombe); ADCK3; ARCA2; CABC1; COQ8; MGC4849; SCAR9
KINOMEscan Wild Type; Full length
200047 AXL 200047 P30530
AXL receptor tyrosine kinase; AXL; JTK11; UFO
KINOMEscan Wild Type; Partial length
200046 AURKC 200046 Q9UQB9
Aurora kinase C; AIE2; AIK3; ARK3; Aur3; AurC; AurC/Aur3; AURKC; aurora-C; STK13
KINOMEscan Wild Type; Full length
200031 ACVRL1 200031 P37023
Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
KINOMEscan Wild Type; Partial length
200045 AURKB 200045 Q96GD4
Aurora kinase B; AIK2; AIM1; AIM-1; ARK2; Aur1; AurB; AurB/Aur1; AURKB; aurkb-sv1; aurkb-sv2; IPL1; STK12; STK5
KINOMEscan Wild Type; Partial length
200044 AURKA 200044 O14965
Aurora kinase A; AIK; AIRK1; ARK1; Aur2; AURA; AurA/Aur2; AURKA; AURORA2; Aurora-A; Ayk1; BTAK; IAK; IAK1; MGC34538; STK15; STK6; STK7
KINOMEscan Wild Type; Partial length
200042 M3K5 200042 Q99683
Mitogen-activated protein kinase kinase kinase 5; ASK; ASK/MAP3K5; ASK1; MAP3K5; MAPKKK5; MEKK5
KINOMEscan Wild Type; Partial length
200067 KCC4 200067 Q16566
Calcium/calmodulin-dependent protein kinase type IV; CAMK4; CaMK-GR; MGC36771
KINOMEscan Wild Type; Partial length
200041 NUAK1 200041 O60285
NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1
KINOMEscan Wild Type; Partial length
200030 ACVR2B 200030 Q13705
Activin A receptor, type IIB; ActR2B; ACTRIIB; ActR-IIB; ACVR2B; MGC116908
KINOMEscan Wild Type; Partial length
200029 ACVR2A 200029 P27037
Activin A receptor, type IIA; ActR2; ACTRII; ACVR2; ACVR2A
KINOMEscan Wild Type; Partial length
200065 KCC2D 200065 Q13557
Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911
KINOMEscan Wild Type; Partial length
200040 ANKK1 200040 Q8NFD2
Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288
KINOMEscan Wild Type; Partial length
200064 CAMK2B 200064 Q13554
Calcium/calmodulin-dependent protein kinase II beta; CAM2; CAMK2; CAMK2B; CAMKB; MGC29528
KINOMEscan Wild Type; Partial length
200063 CAMK2A 200063 Q9UQM7
Calcium/calmodulin-dependent protein kinase II alpha; CAMK2A; CAMKA; KIAA0968
KINOMEscan Wild Type; Partial length
200066 CAMK2G 200066 Q13555
Calcium/calmodulin-dependent protein kinase II gamma; CAMK; CAMK2G; CAMKG; CAMK-II; FLJ16043; MGC26678
KINOMEscan Wild Type; Partial length
200039 AMPK-alpha2 200039 P54646
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2
KINOMEscan Wild Type; Partial length
200068 KKCC1 200068 Q8N5S9
Calcium/calmodulin-dependent protein kinase kinase 1, CaM-kinase IV kinase; CAMKK1; CAMKKA; DKFZp761M0423; MGC34095
KINOMEscan Wild Type; Partial length
200028 ACVR1B 200028 P36896
Activin A receptor, type IB; ACTRIB; ACVR1B; ACVRLK4; ALK4; SKR2
KINOMEscan Wild Type; Partial length
200062 CAMK1G 200062 Q96NX5
Calcium/calmodulin-dependent protein kinase IG; CAMK1G; CLICKIII; dJ272L16.1; VWS1
KINOMEscan Wild Type; Partial length