NU7441 KINOMEscan - Dataset (ID:20040)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200034 AKT1 200034 P31749
V-akt murine thymoma viral oncogene homolog 1; AKT; AKT1; Akt1/PKBa; MGC99656; PKB; PKBa; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA
KINOMEscan Wild Type; Partial length
200035 AKT2 200035 P31751
V-akt murine thymoma viral oncogene homolog 2; AKT2; Akt2/PKBb; PKBb; PKBBETA; PRKBB; RAC-BETA
KINOMEscan Wild Type; Partial length
200181 GRK4 200181 P32298
G protein-coupled receptor kinase 4; GPRK2L; GPRK4; GRK4; GRK4a; IT11
KINOMEscan Wild Type; Full length
200448 TTK 200448 P33981
TTK protein kinase; CT96; ESK; FLJ38280; MPS1; MPS1L1; PYT; TTK
KINOMEscan Wild Type; Partial length
200435 TIE1 200435 P35590
Tyrosine-protein kinase receptor Tie-1; tyrosine kinase with immunoglobulin-like and EGF-like domains 1; JTK14; TIE; TIE1
KINOMEscan Wild Type; Partial length
200175 FLT4 200175 P35916
Fms-related tyrosine kinase 4; FLT4; FLT41; LMPH1A; PCL; VEGFR3
KINOMEscan Wild Type; Partial length
200458 VGFR2 200458 P35968
Vascular endothelial growth factor receptor 2; kinase insert domain receptor; CD309; FLK1; FLK-1; KDR; KRD-1; Ly73; VEGFR; VEGFR2; VEGFR-2
KINOMEscan Wild Type; Partial length
200252 MP2K2 200252 P36507
Dual specificity mitogen-activated protein kinase kinase 2; mitogen-activated protein kinase kinase 2; FLJ26075; MAP2K2; MAPKK2; MEK2; MEK2/MAP2K2; MKK2; PRKMK2
KINOMEscan Wild Type; Full length
200174 FLT3(R834Q) 200174 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan R834Q Mutation (R834Q); Partial length
200173 FLT3(N841I) 200173 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan N841I Mutation (N841I); Partial length
200172 FLT3(K663Q) 200172 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan K663Q Mutation (K663Q); Partial length
200171 FLT3(ITD) 200171 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan ITD Mutation (ITD); Partial length
200170 FLT3(D835Y) 200170 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan D835Y Mutation (D835Y); Partial length
200169 FLT3(D835H) 200169 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan D835H Mutation (D835H); Partial length
200168 FLT3 200168 P36888
Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1
KINOMEscan Wild Type; Partial length
200050 BMPR1A 200050 P36894
Bone morphogenetic protein receptor, type IA; 10q23del; ACVRLK3; ALK3; BMPR1A; CD292; SKR5
KINOMEscan Wild Type; Partial length
200028 ACVR1B 200028 P36896
Activin A receptor, type IB; ACTRIB; ACVR1B; ACVRLK4; ALK4; SKR2
KINOMEscan Wild Type; Partial length
200433 TGFBR1 200433 P36897
Transforming growth factor, beta receptor 1; AAT5; ACVRLK4; ALK5; ALK-5; LDS1A; LDS2A; SKR4; TGFBR1; TGFR-1
KINOMEscan Wild Type; Partial length
200031 ACVRL1 200031 P37023
Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
KINOMEscan Wild Type; Partial length
200434 TGFBR2 200434 P37173
Transforming growth factor, beta receptor II (70/80kDa); AAT3; FAA3; LDS1B; LDS2B; MFS2; RIIC; TAAD2; TGFbeta-RII; TGFBR2; TGFR-2
KINOMEscan Wild Type; Partial length
200095 CSK 200095 P41240
C-src tyrosine kinase; CSK; MGC117393
KINOMEscan Wild Type; Full length
200357 KPCI 200357 P41743
Protein kinase C, iota; DXS1179E; MGC26534; nPKC-iota; PKCI; PRKCI
KINOMEscan Wild Type; Partial length
200327 PIK3CA(E545K) 200327 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E545K Mutation (E545K); Partial length
200324 PIK3CA(C420R) 200324 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan C420R Mutation (C420R); Partial length
200325 PIK3CA(E542K) 200325 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E542K Mutation (E542K); Partial length