AZ-628 KINOMEscan - Dataset (ID:20025)
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| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| AZ-628 | ABL2 | 12.0 | 10 | uM |
| AZ-628 | ABL1(Y253F)-phosphorylated | 1.4 | 10 | uM |
| AZ-628 | ABL1(T315I)-phosphorylated | 79.0 | 10 | uM |
| AZ-628 | ABL1(T315I)-nonphosphorylated | 49.0 | 10 | uM |
| AZ-628 | ABL1(Q252H)-phosphorylated | 3.0 | 10 | uM |
| AZ-628 | ABL1(Q252H)-nonphosphorylated | 2.2 | 10 | uM |
| AZ-628 | ABL1-phosphorylated | 1.4 | 10 | uM |
| AZ-628 | ABL1-nonphosphorylated | 0.1 | 10 | uM |
| AZ-628 | ABL1(M351T)-phosphorylated | 3.3 | 10 | uM |
| AZ-628 | ABL1(H396P)-phosphorylated | 2.6 | 10 | uM |
| AZ-628 | ABL1(H396P)-nonphosphorylated | 0.4 | 10 | uM |
| AZ-628 | ABL1(F317L)-phosphorylated | 6.4 | 10 | uM |
| AZ-628 | ABL1(F317L)-nonphosphorylated | 4.6 | 10 | uM |
| AZ-628 | ABL1(F317I)-phosphorylated | 26.0 | 10 | uM |
| AZ-628 | ABL1(F317I)-nonphosphorylated | 7.3 | 10 | uM |
| AZ-628 | ABL1(E255K)-phosphorylated | 3.4 | 10 | uM |
| AZ-628 | AAK1 | 100.0 | 10 | uM |