Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
Alisertib
9475
3
ROCK2
Alisertib
9448
3
MAP4K4
Alisertib
8550
3
MAPKAPK5
Alisertib
9263
3
STK17A
Alisertib
3717
3
JAK2
Alisertib
1452
3
CSNK1A1
Alisertib
9261
3
MAPKAPK2
Alisertib
2444
2
FRK
Alisertib
1020
3
CDK5
ALK-IN-1
1956
2
EGFR
ALK-IN-1
6098
1
ROS1
ALK-IN-1
238
1
ALK
Alpelisib
1760
10
DMPK
Alpelisib
5287
10
PIK3C2B
Alpelisib
65267
10
WNK3
Alpelisib
65125
10
WNK1
Alpelisib
2045
10
EPHA7
Alpelisib
65061
10
CDK15
Alpelisib
65266
10
WNK4
Alpelisib
208
10
AKT2
Alpelisib
5593
10
PRKG2
Alpelisib
57787
10
MARK4
Alpelisib
65268
10
WNK2
Alpelisib
57551
10
TAOK1
Alpelisib
4067
10
LYN