Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
Disulfiram
216
2
ALDH1A1
Disulfiram
8854
2
ALDH1A2
Disulfiram
219
2
ALDH1B1
Disulfiram
29539
10
Aldh2
Disulfiram
217
2
ALDH2
Disulfiram
221
2
ALDH3B1
Disulfiram
222
2
ALDH3B2
GNF-5837
11682
3
Alk
NVP-TAE684
11682
1
Alk
NVP-TAE684
11682
1
Alk
Seliciclib
238
3
ALK
ALW-II-38-3
238
10
ALK
GSK1838705A
238
1
ALK
Alpelisib
238
10
ALK
Afatinib
238
10
ALK
Cediranib
238
3
ALK
SB202190
238
3
ALK
Axitinib
238
3
ALK
Sotrastaurin
238
3
ALK
Barasertib
238
3
ALK
Ellagic acid
238
10
ALK
PP1
238
3
ALK
GW2580
238
10
ALK
Ceritinib
238
1
ALK
ALK-IN-1
238
1
ALK