Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
Pazopanib
102724428
3
SIK1B
Pazopanib
102724428
3
SIK1B
Pazopanib
102724428
3
SIK1B
Canertinib
102724428
10
SIK1B
Canertinib
102724428
10
SIK1B
Ibrutinib
102724428
10
SIK1B
Fedratinib
102724428
1
SIK1B
Fedratinib
102724428
1
SIK1B
Omipalisib
102724428
10
SIK1B
Buparlisib
102724428
10
SIK1B
Nintedanib
102724428
2
SIK1B
Nintedanib
102724428
2
SIK1B
Foretinib
102724428
2
SIK1B
Foretinib
102724428
2
SIK1B
SP600125
102724428
10
SIK1B
TGX221
102724428
10
SIK1B
GSK1059615
102724428
10
SIK1B
Sunitinib
102724428
3
SIK1B
Sunitinib
102724428
3
SIK1B
Sunitinib
102724428
3
SIK1B
BGJ398
102724428
10
SIK1B
Bosutinib
102724428
1
SIK1B
Bosutinib
102724428
1
SIK1B
KW2449
102724428
2
SIK1B
KW2449
102724428
2
SIK1B