Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
KIN001-127
25
10
ABL1
A443654
25
10
ABL1
Pictilisib
25
10
ABL1
Pictilisib
25
10
ABL1
PD184352
25
10
ABL1
PD184352
25
10
ABL1
PLX-4720
25
3
ABL1
PLX-4720
25
3
ABL1
Lapatinib
25
10
ABL1
Lapatinib
25
10
ABL1
ZSTK474
25
10
ABL1
Selumetinib
25
10
ABL1
Selumetinib
25
10
ABL1
AZD-6482
25
10
ABL1
TAK-715
25
2
ABL1
NU7441
25
10
ABL1
WYE-125132
25
10
ABL1
MLN8054
25
2
ABL1
MLN8054
25
2
ABL1
Barasertib
25
3
ABL1
Barasertib
25
3
ABL1
Enzastaurin
25
10
ABL1
Enzastaurin
25
10
ABL1
NPK76-II-72-1
25
10
ABL1
Palbociclib
25
3
ABL1