Abemaciclib KINOMEscan - Dataset - HMS LINCS Database

Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small molecules	Proteins

Small Molecule	Protein	% Control	Assay compound conc	Conc unit
Abemaciclib	AAK1	20.0	100	nM
Abemaciclib	AAK1	2.0	1000	nM
Abemaciclib	ABL1(E255K)-phosphorylated	81.0	100	nM
Abemaciclib	ABL1(E255K)-phosphorylated	82.0	1000	nM
Abemaciclib	ABL1(F317I)-nonphosphorylated	100.0	100	nM
Abemaciclib	ABL1(F317I)-nonphosphorylated	100.0	1000	nM
Abemaciclib	ABL1(F317I)-phosphorylated	91.0	100	nM
Abemaciclib	ABL1(F317I)-phosphorylated	100.0	1000	nM
Abemaciclib	ABL1(F317L)-nonphosphorylated	99.0	100	nM
Abemaciclib	ABL1(F317L)-nonphosphorylated	86.0	1000	nM
Abemaciclib	ABL1(F317L)-phosphorylated	100.0	100	nM
Abemaciclib	ABL1(F317L)-phosphorylated	100.0	1000	nM
Abemaciclib	ABL1(H396P)-nonphosphorylated	80.0	100	nM
Abemaciclib	ABL1(H396P)-nonphosphorylated	56.0	1000	nM
Abemaciclib	ABL1(H396P)-phosphorylated	89.0	100	nM
Abemaciclib	ABL1(H396P)-phosphorylated	96.0	1000	nM
Abemaciclib	ABL1(M351T)-phosphorylated	100.0	100	nM
Abemaciclib	ABL1(M351T)-phosphorylated	100.0	1000	nM
Abemaciclib	ABL1(Q252H)-nonphosphorylated	80.0	100	nM
Abemaciclib	ABL1(Q252H)-nonphosphorylated	50.0	1000	nM
Abemaciclib	ABL1(Q252H)-phosphorylated	97.0	100	nM
Abemaciclib	ABL1(Q252H)-phosphorylated	100.0	1000	nM
Abemaciclib	ABL1(T315I)-nonphosphorylated	20.0	100	nM
Abemaciclib	ABL1(T315I)-nonphosphorylated	0.0	1000	nM
Abemaciclib	ABL1(T315I)-phosphorylated	97.0	100	nM