LY-317615 KINOMEscan - Dataset (ID:20159)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Enzastaurin | DCAMKL2 | nM | |
Enzastaurin | DCAMKL3 | nM | |
Enzastaurin | DDR1 | nM | |
Enzastaurin | DDR2 | nM | |
Enzastaurin | M3K12 | nM | |
Enzastaurin | DMPK | 2200.0 | nM |
Enzastaurin | DMPK2 | nM | |
Enzastaurin | DRAK1 | 760.0 | nM |
Enzastaurin | DRAK2 | nM | |
Enzastaurin | DYRK1A | 160.0 | nM |
Enzastaurin | DYRK1B | 1000.0 | nM |
Enzastaurin | DYRK2 | nM | |
Enzastaurin | EGFR | nM | |
Enzastaurin | EGFR(E746-A750del) | nM | |
Enzastaurin | EGFR(G719C) | nM | |
Enzastaurin | EGFR(G719S) | nM | |
Enzastaurin | EGFR(L747-E749del, A750P) | nM | |
Enzastaurin | EGFR(L747-S752del, P753S) | nM | |
Enzastaurin | EGFR(L747-T751del,Sins) | nM | |
Enzastaurin | EGFR(L858R) | nM | |
Enzastaurin | EGFR(L858R,T790M) | nM | |
Enzastaurin | EGFR(L861Q) | nM | |
Enzastaurin | EGFR(S752-I759del) | nM | |
Enzastaurin | EGFR(T790M) | nM | |
Enzastaurin | EIF2AK1 | nM |