Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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  • Page 1 of 18
  • 1 to 25 of 432 records
Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
HCC1806 XL147 3 72
flat
flat
HCC1806 pilaralisib 0 3 72
8 3.185
Inf
1.02
0.000871
0.0
1.02
0.01
-2.12e-06
1.0
1.0
Inf
1.03
0.999
0.0
1.03
0.01
-0.000107
1.0
1.0
HCC1806 XL147 1 72
flat
flat
HCC1806 pilaralisib 0 1 72
8 2.732
Inf
1.02
0.00101
0.0
1.02
0.01
-4.53e-06
1.0
1.0
Inf
1.03
0.999
0.0
1.03
0.01
-0.000107
1.0
1.0
HCC1806 XL147 2 72
flat
flat
HCC1806 pilaralisib 0 2 72
8 2.817
Inf
1.02
0.000975
0.0
1.02
0.01
-4.46e-06
1.0
1.0
Inf
1.03
0.999
0.0
1.03
0.01
-0.000109
1.0
1.0
BT-549 XL147 2 72
flat
flat
BT549 pilaralisib 0 2 72
8 1.952
Inf
0.967
-0.00824
0.0
0.967
0.01
-0.000427
1.0
1.0
Inf
0.968
1.01
0.0
0.968
0.01
-0.000878
1.0
1.0
HCC1806 AZD-6482 2 72
flat
flat
HCC1806 AZD6482 0 2 72
8 2.833
Inf
1.0
0.00136
0.0
1.0
0.01
-0.0062
1.0
0.999
Inf
1.01
0.998
0.0
1.01
0.01
-0.00512
1.0
0.998
HCC1806 AZD-6482 1 72
flat
flat
HCC1806 AZD6482 0 1 72
8 2.748
Inf
1.0
0.00141
0.0
1.0
0.01
-0.00621
1.0
0.999
Inf
1.01
0.998
0.0
1.01
0.01
-0.00515
1.0
0.998
HCC1806 AZD-6482 3 72
flat
flat
HCC1806 AZD6482 0 3 72
8 3.201
Inf
1.0
0.00122
0.0
1.0
0.01
-0.0063
1.0
0.999
Inf
1.01
0.998
0.0
1.01
0.01
-0.00515
1.0
0.998
HCC70 Alpelisib 2 72
flat
flat
HCC70 alpelisib 0 2 72
8 1.799
Inf
0.748
0.0777
0.0
0.748
0.01
0.00864
0.974
0.907
Inf
0.785
0.932
0.0
0.785
0.01
0.00534
0.984
0.919
BT-20 BX-912 3 72
flat
flat
BT20 BX-912 0 3 72
8 2.619
Inf
0.904
0.0795
0.0
0.904
0.01
0.000173
0.999
0.918
Inf
0.879
0.9
0.0
0.879
0.01
0.00619
0.982
0.896
BT-20 XL147 2 72
flat
flat
BT20 pilaralisib 0 2 72
8 1.784
Inf
0.759
0.073
0.0
0.759
0.01
-0.0058
1.0
0.907
Inf
0.796
0.937
0.0
0.796
0.01
-0.00637
1.0
0.92
BT-20 KIN001-244 1 72
flat
flat
BT20 KIN001-244 0 1 72
8 2.125
Inf
0.911
0.0401
0.0
0.911
0.01
-0.00641
1.0
0.957
Inf
0.908
0.958
0.0
0.908
0.01
-0.00745
1.0
0.955
BT-20 TGX221 1 72
flat
flat
BT20 TGX-221 0 1 72
8 1.988
Inf
1.02
-0.00357
0.0
1.02
0.01
-0.00762
1.0
1.0
Inf
1.02
1.0
0.0
1.02
0.01
-0.00881
1.0
1.0
HCC70 KIN001-244 3 72
flat
flat
HCC70 KIN001-244 0 3 72
8 2.472
Inf
0.916
0.0295
0.0
0.916
0.01
-0.0208
1.0
0.969
Inf
0.899
0.965
0.0
0.899
0.01
-0.00883
1.0
0.963
BT-549 Alpelisib 3 72
flat
flat
BT549 alpelisib 0 3 72
8 1.743
Inf
0.817
0.068
0.0
0.817
0.01
-0.0192
1.0
0.915
Inf
0.846
0.942
0.0
0.846
0.01
-0.0162
1.0
0.928
HCC38 KIN001-244 2 72
flat
flat
HCC38 KIN001-244 0 2 72
8 2.210
Inf
0.948
0.0304
0.0
0.948
0.01
-0.0213
1.0
0.969
Inf
0.944
0.967
0.0
0.944
0.01
-0.0218
1.0
0.966
HCC38 Alpelisib 2 72
flat
flat
HCC38 alpelisib 0 2 72
8 2.086
Inf
0.848
0.0559
0.0
0.848
0.01
-0.0371
1.0
0.931
Inf
0.848
0.944
0.0
0.848
0.01
-0.0359
1.0
0.932
HCC38 XL147 2 72
flat
flat
HCC38 pilaralisib 0 2 72
8 2.194
Inf
0.938
0.0288
0.0
0.938
0.01
-0.0925
1.0
0.968
Inf
0.933
0.969
0.0
0.933
0.01
-0.0418
1.0
0.965
HCC70 KIN001-244 2 72
flat
flat
HCC70 KIN001-244 0 2 72
8 1.684
Inf
0.898
-0.0201
0.0
0.898
0.01
0.508
0.119
1.01
Inf
0.916
1.02
0.0
0.916
0.01
-0.0458
1.0
1.01
BT-20 XL147 3 72
flat
flat
BT20 pilaralisib 0 3 72
8 2.647
Inf
0.755
0.102
0.0
0.755
0.01
0.0679
0.81
0.885
Inf
0.708
0.871
0.0
0.708
0.01
0.0505
0.856
0.857
BT-20 CAL-101 3 72
flat
flat
BT20 idelalisib 0 3 72
8 2.589
Inf
0.916
0.0535
0.0
0.916
0.01
0.0547
0.845
0.944
Inf
0.894
0.932
0.0
0.894
0.01
0.0506
0.856
0.929
BT-20 TGX221 3 72
flat
flat
BT20 TGX-221 0 3 72
8 2.469
Inf
1.01
0.0147
0.0
1.01
0.01
-0.0563
1.0
0.982
Inf
1.01
0.983
0.0
1.01
0.01
-0.0552
1.0
0.979
HCC1806 KIN001-244 3 72
flat
flat
HCC1806 KIN001-244 0 3 72
8 3.195
Inf
0.988
0.0203
0.0
0.988
0.01
-0.0575
1.0
0.982
Inf
0.981
0.968
0.0
0.981
0.01
-0.0553
1.0
0.972
HCC1806 KIN001-244 2 72
flat
flat
HCC1806 KIN001-244 0 2 72
8 2.827
Inf
0.986
0.0229
0.0
0.986
0.01
-0.0574
1.0
0.98
Inf
0.981
0.968
0.0
0.981
0.01
-0.0553
1.0
0.972
HCC1806 KIN001-244 1 72
flat
flat
HCC1806 KIN001-244 0 1 72
8 2.742
Inf
0.986
0.0236
0.0
0.986
0.01
-0.0573
1.0
0.979
Inf
0.981
0.968
0.0
0.981
0.01
-0.0553
1.0
0.972
HCC38 XL147 1 72
flat
flat
HCC38 pilaralisib 0 1 72
8 1.752
Inf
0.949
0.0257
0.0
0.949
0.01
-0.0703
1.0
0.973
Inf
0.955
0.978
0.0
0.955
0.01
-0.0701
1.0
0.977
  • Page 1 of 18
  • 1 to 25 of 432 records