Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
COLO 858 Vemurafenib GSK-J1 0.3160 2.6667
uM
48
hr
1 1988 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 344.25 NGFR rabbit IgG(H+L) / donkey NGFR 140.14
Colo858-A2-rep1
B6
COLO 858 Vemurafenib (+)-JQ1 0.3160 2.6667
uM
48
hr
1 1745 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.39 NGFR rabbit IgG(H+L) / donkey NGFR 10.46
Colo858-A2-rep1
C7
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 920 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 297.13 NGFR rabbit IgG(H+L) / donkey NGFR 146.65
Colo858-A2-rep1
A6
COLO 858 Vemurafenib Rocilinostat 0.3160 2.6667
uM
48
hr
1 755 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 163.81 NGFR rabbit IgG(H+L) / donkey NGFR 184.22
Colo858-A2-rep1
B5
COLO 858 Vemurafenib Rucaparib 0.3160 2.6667
uM
48
hr
1 2594 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 255.48 NGFR rabbit IgG(H+L) / donkey NGFR 179.23
Colo858-A2-rep1
C3
COLO 858 Vemurafenib GSK-J2 0.3160 2.6667
uM
48
hr
1 2652 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 335.90 NGFR rabbit IgG(H+L) / donkey NGFR 155.80
Colo858-A2-rep1
C6
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1202 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 347.86 NGFR rabbit IgG(H+L) / donkey NGFR 141.29
Colo858-A2-rep1
A2
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1122 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 296.79 NGFR rabbit IgG(H+L) / donkey NGFR 157.80
Colo858-A2-rep1
A5
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1371 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 358.01 NGFR rabbit IgG(H+L) / donkey NGFR 148.58
Colo858-A2-rep1
A9
COLO 858 Vemurafenib CTB 0.3160 2.6667
uM
48
hr
1 1748 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 291.14 NGFR rabbit IgG(H+L) / donkey NGFR 149.16
Colo858-A2-rep1
B4
COLO 858 Vemurafenib UNC669 0.3160 2.6667
uM
48
hr
1 2097 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 357.07 NGFR rabbit IgG(H+L) / donkey NGFR 157.23
Colo858-A2-rep1
B8
COLO 858 Vemurafenib Veliparib 0.3160 2.6667
uM
48
hr
1 2017 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 297.02 NGFR rabbit IgG(H+L) / donkey NGFR 148.72
Colo858-A2-rep1
C2
COLO 858 Vemurafenib Belinostat 0.3160 2.6667
uM
48
hr
1 209 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 309.25 NGFR rabbit IgG(H+L) / donkey NGFR 21.49
Colo858-A2-rep1
C4
COLO 858 Vemurafenib Selisistat 0.3160 2.6667
uM
48
hr
1 3015 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 359.72 NGFR rabbit IgG(H+L) / donkey NGFR 105.69
Colo858-A2-rep1
C5
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1391 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 358.32 NGFR rabbit IgG(H+L) / donkey NGFR 158.87
Colo858-A2-rep1
A10
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1242 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 296.85 NGFR rabbit IgG(H+L) / donkey NGFR 156.51
Colo858-A2-rep1
A11
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1024 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 345.50 NGFR rabbit IgG(H+L) / donkey NGFR 135.78
Colo858-A2-rep1
A3
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1076 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 288.18 NGFR rabbit IgG(H+L) / donkey NGFR 162.29
Colo858-A2-rep1
A4
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 1095 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 337.39 NGFR rabbit IgG(H+L) / donkey NGFR 164.33
Colo858-A2-rep1
A7
COLO 858 Vemurafenib 0.3160
uM
48
hr
1 897 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 335.21 NGFR rabbit IgG(H+L) / donkey NGFR 126.80
Colo858-A2-rep1
A8
COLO 858 Vemurafenib Olaparib 0.3160 2.6667
uM
48
hr
1 1345 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 290.82 NGFR rabbit IgG(H+L) / donkey NGFR 146.21
Colo858-A2-rep1
B2
COLO 858 Vemurafenib Iniparib 0.3160 2.6667
uM
48
hr
1 1703 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 310.30 NGFR rabbit IgG(H+L) / donkey NGFR 122.97
Colo858-A2-rep1
B3
COLO 858 Vemurafenib PFI-1 0.3160 2.6667
uM
48
hr
1 1383 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 138.34 NGFR rabbit IgG(H+L) / donkey NGFR 30.41
Colo858-A2-rep1
B7
COLO 858 Vemurafenib Vorinostat 0.3160 2.6667
uM
48
hr
1 329 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 200.63 NGFR rabbit IgG(H+L) / donkey NGFR 17.50
Colo858-A2-rep1
D2
COLO 858 Vemurafenib UNC1215 0.3160 2.6667
uM
48
hr
1 2700 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 375.51 NGFR rabbit IgG(H+L) / donkey NGFR 134.85
Colo858-A2-rep1
C8
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