Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 2 of 4: Calculated dose-response metrics. - Dataset (ID:20269)

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Cell Clinical Subtype Transcriptional Subtype Small Molecule Antibody Perturbagen Target Perturbagen Class Biological Replicate ID Conc Unit GR50 GEC50 GRmax GRinf GR Hill Coefficient GR_AOC GR r2 Nominal Division Rate
HCC1187
TNBC
Basal A
Epirubicin
TOP2
TOP
7811.017
uM
0.08798
0.25888
-1.0000 -1.0000 1.0180 1.0515
0.9521
0.3604
HCC1395
TNBC
Basal B
GSK1070916
AURK
AURK
9254.001
uM
5.38610
6.70950
-1.0000 -0.9998 5.0000 0.3079
0.9082
0.3986
HCC1187
TNBC
Basal A
17-AAG
HSP90
HSP90
7811.04
uM
1.04690
1.38930
-1.0000 -0.9258 3.7023 0.7792
0.8482
0.3921
HCC1187
TNBC
Basal A
Cisplatin
DNA cross-linker
DNA cross-linker
9244.021
uM
2.02180
2.59060
-1.0000 -0.9970 4.4235 0.7319
0.9785
0.4542
HCC1395
TNBC
Basal B
CGC-11047
Polyamine analogue
9258.026
uM
0.44087
35.50130
-1.0000 -1.0000 0.2503 0.8247
0.7494
0.5632
HCC1395
TNBC
Basal B
Cisplatin
DNA cross-linker
DNA cross-linker
9258.03
uM
1.05110
2.06760
-1.0000 -1.0000 1.6238 0.7227
0.9985
0.4015
BT-20
TNBC
Basal A
MG-132
Proteasome
Proteasome
14230.189
uM
0.13122
0.14986
-1.0000 -0.4715 5.0000 0.7755
0.5873
0.4635
HCC1187
TNBC
Basal A
(Z)-4-Hydroxytamoxifen
ESR1
7811.044
uM
11.65150
16.05880
-1.0000 -0.9995 3.4233 0.3459
0.9975
0.3073
BT-474
HER2amp
Luminal
Gefitinib
EGFR
ErbB
9158.049
uM
1.82990
2.5510
-1.0000 -0.9995 3.3059 0.5005
0.9072
0.4082
HCC1187
TNBC
Basal A
Cisplatin
DNA cross-linker
DNA cross-linker
7811.017
uM
1.68090
2.53690
-1.0000 -1.0000 2.6690 0.9047
0.7309
0.3604
HCC1187
TNBC
Basal A
Methylglyoxal
13726.184
uM
0.99124
16.40040
-1.0000 -1.0000 0.3915 1.2606
0.7991
0.3574
HCC1187
TNBC
Basal A
Oxaliplatin
DNA cross-linker
DNA cross-linker
7811.011
uM
0.26894
0.77535
-1.0000 -1.0000 1.0376 1.1173
0.9558
0.4400
BT-474
HER2amp
Luminal
CGC-11047
Polyamine analogue
9163.026
uM
1.16670
17.90580
-1.0000 -1.0000 0.4023 0.8897
0.9004
0.3738
BT-474
HER2amp
Luminal
Bromopyruvic acid
Hexokinase II
Metabolism
13125.177
uM
0.37090
0.53838
-1.0000 -0.9928 2.9354 0.6307
0.9967
0.8991
600MPE
HR+
Luminal
Bromopyruvic acid
Hexokinase II
Metabolism
13091.177
uM
0.13548
0.2280
-1.0000 -1.0000 2.1106 0.8509
0.9450
0.7004
184B5
NM
Basal
Bromopyruvic acid
Hexokinase II
Metabolism
12979.177
uM
0.02740
0.03413
-1.0000 -1.0000 5.0000 1.0789
0.9988
0.5647
BT-20
TNBC
Basal A
Z-Leu-Leu-Norvalinal
Proteasome
Proteasome
14230.189
uM
0.27401
0.47494
-1.0000 -1.0000 1.9974 0.7978
0.9974
0.4635
184B5
NM
Basal
Chloroquine
12979.177
uM
19.64650
24.47430
-1.0000 -1.0000 5.0000 0.1512
0.9526
0.5647
BT-474
HER2amp
Luminal
Doxorubicin
TOP2
TOP
9163.121
uM
0.18301
0.22105
-1.0000 -0.7856 5.0000 0.7812
0.9752
0.4382
BT-20
TNBC
Basal A
MG-132
Proteasome
Proteasome
14230.189
uM
0.13122
0.14986
-1.0000 -0.4715 5.0000 0.7755
0.5873
0.4635
AU565
HER2amp
Luminal
Methylglyoxal
13030.184
uM
50.30640
183.32630
-1.0000 -1.0000 0.8496 0.9024
0.9717
0.5725
600MPE
HR+
Luminal
Chloroquine
13091.177
uM
inf
inf
-1.0000 -1.0000 0.0000 0.3682
0.5443
0.7004
184A1
NM
Basal
Doxorubicin
TOP2
TOP
10002.034
uM
0.10668
0.20741
-1.0000 -0.9682 1.6201 0.9516
0.9936
0.6736
HCC1395
TNBC
Basal B
GSK461364
PLK1
PLK
9254.001
uM
0.00450
0.00522
-1.0000 -0.5435 5.0000 1.0717
0.8911
0.3986
HCC1395
TNBC
Basal B
GSK1838705A
IGF1R
RTK
7435.091
uM
3.60990
6.22790
-1.0000 -1.0000 2.0145 0.5103
0.9880
0.5716
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