Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib ACVR2A 99.0 100
nM
Taselisib ADCK4 100.0 100
nM
Taselisib ABL1-phosphorylated 91.0 100
nM
Taselisib ACVR1B 99.0 100
nM
Taselisib ACVRL1 100.0 100
nM
Taselisib ADCK3 100.0 100
nM
Taselisib ABL1(Y253F)-phosphorylated 96.0 100
nM
Taselisib ABL1-nonphosphorylated 88.0 100
nM
Taselisib ABL2 94.0 100
nM
Taselisib ACVR1 100.0 100
nM
Taselisib ACVR2B 92.0 100
nM
Taselisib ABL1(H396P)-nonphosphorylated 79.0 100
nM
Taselisib ABL1(F317I)-phosphorylated 78.0 100
nM
Taselisib ABL1(H396P)-phosphorylated 80.0 100
nM
Taselisib AAK1 77.0 100
nM
Taselisib ABL1(M351T)-phosphorylated 94.0 100
nM
Taselisib ABL1(F317L)-nonphosphorylated 90.0 100
nM
Taselisib ABL1(Q252H)-nonphosphorylated 87.0 100
nM
Taselisib ABL1(F317I)-nonphosphorylated 88.0 100
nM
Taselisib ABL1(Q252H)-phosphorylated 80.0 100
nM
Taselisib ABL1(F317L)-phosphorylated 100.0 100
nM
Taselisib ABL1(T315I)-nonphosphorylated 85.0 100
nM
Taselisib ABL1(E255K)-phosphorylated 75.0 100
nM
Taselisib ABL1(T315I)-phosphorylated 100.0 100
nM
Taselisib AKT1 92.0 100
nM
  • Page 1 of 38
  • 1 to 25 of 936 records